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MLS-573151

Catalog No. T22106 CAS 10179-57-4

MLS-573151 is a selective inhibitor of GTPase Cdc42(EC50 of 2 μM). It is inactive against other GTPases family members, such as Rab2, Rab7, H-Ras, Rac1, Rac 2 and RhoA wild-type. MLS-573151 acts by blocking the binding of GTP to Cdc42.

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MLS-573151, CAS 10179-57-4

Pack Size	Availability	Price/USD
1 mg	In stock	$ 34.00
2 mg	In stock	$ 48.00
5 mg	In stock	$ 80.00
10 mg	In stock	$ 139.00
25 mg	In stock	$ 289.00
50 mg	In stock	$ 455.00
100 mg	In stock	$ 672.00
500 mg	In stock	$ 1,430.00
1 mL * 10 mM (in DMSO)	In stock	$ 89.00

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Purity: 99.64%

Biological Description

Chemical Properties

Storage & Solubility Information

Description

Molecular Weight	377.46
Formula	C21H19N3O2S
CAS No.	10179-57-4

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

Solubility Information

DMSO: 30 mg/mL (79.48 mM)

References and Literature

1. Fan Mao, et al. Transcriptomic Evidence Reveals the Molecular Basis for Functional Differentiation of Hemocytes in a Marine Invertebrate, Crassostrea gigas. Front Immunol. 2020 May 27;11:911. 2. Zurab Surviladze, et al. Identification of a small GTPase inhibitor using a high-throughput flow cytometry bead-based multiplex assay. J Biomol Screen. 2010 Jan;15(1):10-20.

Related compound libraries

This product is contained In the following compound libraries：

GPCR Compound Library Inhibitor Library Kinase Inhibitor Library Membrane Protein-targeted Compound Library Bioactive Compound Library Anti-Pancreatic Cancer Compound Library MAPK Inhibitor Library Anti-Liver Cancer Compound Library Anti-Prostate Cancer Compound Library Bioactive Compounds Library Max

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Related compounds with same targets

CDK8-IN-12 VX-11e Purvalanol B CDK12-IN-E9 NU6027 PROTAC CDK9 Degrader-1 AT7519 Hydrochloride MC180295

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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

MLS-573151 10179-57-4 Cell Cycle/Checkpoint GPCR/G Protein MAPK CDK Ras granulocytes Inhibitor inhibit MLS-000573151 MLS 000573151 GTPase Cdc42 MLS000573151 MLS573151 MLS 573151 inhibitor

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