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L 653328

Catalog No. T32458 CAS 115609-61-5

Synonyms: L 653,328, L653328, L653,328, L-653,328, L-653328

L 653328 is an ocular hypotensive agent that has modest beta-receptor blocking activity.

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L 653328, CAS 115609-61-5

Pack Size	Availability	Price/USD
25 mg	6-8 weeks	$ 1,520.00
50 mg	6-8 weeks	$ 1,980.00
100 mg	6-8 weeks	$ 2,500.00

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This compound is a customized synthesis product. We have a strong synthesis team with excellent synthesis technology and capabilities. However, due to various objective factors, there is a low probability that the synthesis will not be successful. If you need to learn more, please feel free to consult us, we will serve you wholeheartedly.

Biological Description

Chemical Properties

Storage & Solubility Information

Description

L 653328 is an ocular hypotensive agent that has modest beta-receptor blocking activity.

Synonyms	L 653,328, L653328, L653,328, L-653,328, L-653328
Molecular Weight	309.4
Formula	C17H27NO4
CAS No.	115609-61-5

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

References and Literature

1. Bauer KG, Brunner-Ferber F, Distlerath LM, Lippa EA, Binkowitz B, Till P, Kaik GA. Assessment of bronchial effects following topical administration of butylamino-phenoxy-propanol-acetate, an oculoselective beta-adrenoceptor blocker in asthmatic subjects. Br J Clin Pharmacol. 1992 Aug;34(2):122-9. PubMed PMID: 1358158; PubMed Central PMCID: PMC1381528. 2. Gerin G, Durand-Cavagna G, Gordon LR, Duprat P, Hollander CF. Drug-induced changes in dogs after long term application of a beta-blocker. Lens Eye Toxic Res. 1989;6(1-2):319-29. PubMed PMID: 2577307. 3. Sugrue MF, Gautheron P, Grove J, Mallorga P, Viader MP, Baldwin JJ, Ponticello GS, Varga SL. L-653,328: an ocular hypotensive agent with modest beta receptor blocking activity. Invest Ophthalmol Vis Sci. 1988 May;29(5):776-84. PubMed PMID: 2896641.

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Method for preparing in vivo formulation：Take μL DMSO master liquid, next add μL PEG300， mix and clarify, next add μL Tween 80，mix and clarify, next add μL ddH₂O, mix and clarify.

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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

L 653328 115609-61-5 L 653,328 L653328 L653,328 L-653,328 L-653328 inhibitor inhibit

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