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K-8012

Catalog No. T24240 CAS 1346513-17-4

Synonyms: K8012, K 8012

K-8012 is a modulator of the N-terminally truncated RXRα and improves anticancer activities in an RXRα-dependent manner.

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K-8012, CAS 1346513-17-4

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Purity: 98%

Biological Description

Chemical Properties

Storage & Solubility Information

Description

K-8012 is a modulator of the N-terminally truncated RXRα and improves anticancer activities in an RXRα-dependent manner.

Synonyms	K8012, K 8012
Molecular Weight	374.463
Formula	C23H23FN4
CAS No.	1346513-17-4

Storage

Powder: -20°C for 3 years

In solvent: -80°C for 2 years

Solubility Information

( < 1 mg/ml refers to the product slightly soluble or insoluble )

References and Literature

1. Chen L, et al. Sulindac-derived RXRα modulators inhibit cancer cell growth by binding to a novel site. Chem Biol. 2014 May 22;21(5):596-607.

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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

K-8012 1346513-17-4 K 8012 K8012 Inhibitor inhibitor inhibit

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