Powder: -20°C for 3 years | In solvent: -80°C for 1 year
GYKI-52466 is a selective non-competitive AMPA receptor antagonist (IC50 values are 10-20, ~ 450 and <50 μM for AMPA-, kainate- and NMDA-induced responses, respectively) used as a Skeletal muscle relaxant, orally active anticonvulsant, neuroprotective and anxiolytic in vivo.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
25 mg | 6-8 weeks | $ 1,520.00 | |
50 mg | 6-8 weeks | $ 1,980.00 | |
100 mg | 6-8 weeks | $ 2,500.00 |
Description | GYKI-52466 is a selective non-competitive AMPA receptor antagonist (IC50 values are 10-20, ~ 450 and >50 μM for AMPA-, kainate- and NMDA-induced responses, respectively) used as a Skeletal muscle relaxant, orally active anticonvulsant, neuroprotective and anxiolytic in vivo. |
Synonyms | GYKI 52,466, GYKI-5,2466, GYKI52,466 |
Molecular Weight | 293.32 |
Formula | C17H15N3O2 |
CAS No. | 102771-26-6 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
H2O: Insoluble
DMSO: Soluble
You can also refer to dose conversion for different animals. More
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GYKI-52466 102771-26-6 GYKI 52,466 GYKI-5,2466 GYKI52466 GYKI52,466 GYKI 52466 inhibitor inhibit