Powder: -20°C for 3 years | In solvent: -80°C for 1 year
TREK1 and TREK2 channel activator (EC50 = 0.76 μM in Rb efflux assay in TREK1-expressing CHO cells). Exhibits selectivity for TREK1/2 over TRAAK, TASK3 and a range of other potassium channels. Hyperpolarizes membrane potential of dorsal root ganglion neurons and depresses neuronal activity in vitro.
Pack Size | Availability | Price/USD | Quantity |
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50 mg | 5 days | Inquiry | |
100 mg | 5 days | Inquiry |
Description | TREK1 and TREK2 channel activator (EC50 = 0.76 μM in Rb efflux assay in TREK1-expressing CHO cells). Exhibits selectivity for TREK1/2 over TRAAK, TASK3 and a range of other potassium channels. Hyperpolarizes membrane potential of dorsal root ganglion neurons and depresses neuronal activity in vitro. |
Molecular Weight | 518.45 |
Formula | C27H20F6N2O2 |
CAS No. | 69563-88-8 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: Soluble
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GI-530159 69563-88-8 GI 530159 GI530159 inhibitor inhibit