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Deramciclane fumarate

Catalog No. T27149 CAS 120444-72-6

Deramciclane fumarate is a 5-HT(2A/C) antagonist with putative anxiolytic activity.

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Deramciclane fumarate Chemical Structure

Deramciclane fumarate, CAS 120444-72-6

Pack Size	Availability	Price/USD
25 mg	6-8 weeks	$ 1,520.00
50 mg	6-8 weeks	$ 1,980.00
100 mg	6-8 weeks	$ 2,500.00

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This compound is a customized synthesis product. We have a strong synthesis team with excellent synthesis technology and capabilities. However, due to various objective factors, there is a low probability that the synthesis will not be successful. If you need to learn more, please feel free to consult us, we will serve you wholeheartedly.

Biological Description

Chemical Properties

Storage & Solubility Information

Description

Deramciclane fumarate is a 5-HT(2A/C) antagonist with putative anxiolytic activity.

Molecular Weight	417.54
Formula	C24H35NO5
CAS No.	120444-72-6

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

References and Literature

1. Kääriäinen TM, Lehtonen M, Forsberg MM, Savolainen J, Käenmäki M, Männistö PT. Comparison of the effects of deramciclane, ritanserin and buspirone on extracellular dopamine and its metabolites in striatum and nucleus accumbens of freely moving rats. Basic Clin Pharmacol Toxicol. 2008 Jan;102(1):50-8. Epub 2007 Oct 25. PubMed PMID: 17971064. 2. Al-Behaisi S, Antal I, Morovján G, Marton S, Klebovich I. The effect of oil as a dietary component on in vitro dissolution of an acid-labile drug. Pharmazie. 2003 Jul;58(7):502-3. PubMed PMID: 12894756. 3. Nemes KB, Abermann M, Bojti E, Grézal G, Al-Behaisi S, Klebovich I. Oral, intraperitoneal and intravenous pharmacokinetics of deramciclane and its N-desmethyl metabolite in the rat. J Pharm Pharmacol. 2000 Jan;52(1):47-51. PubMed PMID: 10716602. 4. Ladányi L, Sztruhár I, Budai Z, Lukács G, Mezei T, Argay G, Kálmán A, Simig G. Stereochemistry and enantiomeric purity of a novel anxiolytic agent, deramciclane fumarate. Chirality. 1999;11(9):689-93. PubMed PMID: 10506429.

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Keywords

Deramciclane fumarate 120444-72-6 Deramciclane Fumarate inhibitor inhibit

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