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Chlorphenesin Carbamate

Catalog No. T21376 CAS 886-74-8

Synonyms: Kolpicortin-sine, Rinlaxer, Chlorphensin carbamate, Maolate, laChlorphenesin Carbamate

Chlorphenesin Carbamate is a centrally acting muscle relaxant used to treat muscle pain and spasms and also an antifungal agent.

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Chlorphenesin Carbamate Chemical Structure

Chlorphenesin Carbamate, CAS 886-74-8

Pack Size	Availability	Price/USD
100 mg	35 days	$ 448.00
250 mg	35 days	$ 1,060.00
500 mg	35 days	$ 1,960.00
1 g	35 days	$ 3,570.00

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Biological Description

Chemical Properties

Storage & Solubility Information

Description

Chlorphenesin Carbamate is a centrally acting muscle relaxant used to treat muscle pain and spasms and also an antifungal agent.

Synonyms	Kolpicortin-sine, Rinlaxer, Chlorphensin carbamate, Maolate, laChlorphenesin Carbamate
Molecular Weight	245.66
Formula	C10H12ClNO4
CAS No.	886-74-8

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

Solubility Information

DMSO: Soluble

H2O: Insoluble

References and Literature

1. Yu JY, Song HH, Kim BG, Park HJ, Choi KS, Kwon YE. Relative bioavailability of generic and branded 250-mg and 500-mg oral chlorphenesin carbamate tablets in healthy Korean volunteers: a single-dose, randomized-sequence, open-label, two-period crossover trial. Clin Ther. 2009 Nov;31(11):2735-43. doi: 10.1016/j.clinthera.2009.11.036. PubMed PMID: 20110015. 2. Okuyama S, Aihara H. Antinociceptive effect of chlorphenesin carbamate in adjuvant arthritic rats. Res Commun Chem Pathol Pharmacol. 1987 Feb;55(2):147-60. PubMed PMID: 3823606. 3. Nozu T, Suwa T, Setoyama K, Kurachi M, Tanaka I. [Influence of the enterohepatic circulation on the metabolism of chlorphenesin carbamate (CPC). I. Comparison between guinea pigs and bile duct-ligated rats (author's transl)]. Yakugaku Zasshi. 1977 Nov;97(11):1189-94. Japanese. PubMed PMID: 616817. 4. Watanabe S, Araki H, Kawasaki H, Ueki S. [Electroencephalographic effects of chlorphenesin carbamate, a new central muscle relaxant, in rabbits (author's transl)]. Nihon Yakurigaku Zasshi. 1977 May;73(4):479-96. Japanese. PubMed PMID: 908544.

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Method for preparing DMSO master liquid: mg drug pre-dissolved in μL DMSO (Master liquid concentration mg/mL)，Please contact us first if the concentration exceeds the DMSO solubility of the batch of drug.

Method for preparing in vivo formulation：Take μL DMSO master liquid, next add μL PEG300， mix and clarify, next add μL Tween 80，mix and clarify, next add μL ddH₂O, mix and clarify.

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What is the mass of compound required to make a 10 mM stock solution in 10 ml of water given that the molecular weight of the compound is 197.13 g/mol?
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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

Chlorphenesin Carbamate 886-74-8 Kolpicortin-sine Rinlaxer Chlorphensin carbamate Maolate laChlorphenesin Carbamate inhibitor inhibit

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