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Carboxypeptidase G2 (CPG2) Inhibitor

Catalog No. T10678 CAS 192203-60-4

Synonyms: Carboxypeptidase G2 Inhibitor, CPG2 Inhibitor

Carboxypeptidase G2 (CPG2) Inhibitor is a new CPG2 Inhibitor with antitumor activity.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

Carboxypeptidase G2 (CPG2) Inhibitor, CAS 192203-60-4

Pack Size	Availability	Price/USD
1 mg	In stock	$ 86.00
5 mg	In stock	$ 208.00
10 mg	In stock	$ 312.00
25 mg	In stock	$ 531.00
50 mg	In stock	$ 768.00
100 mg	In stock	$ 1,070.00
500 mg	In stock	$ 2,150.00

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Purity: 99.69%

Biological Description

Chemical Properties

Storage & Solubility Information

Description

Carboxypeptidase G2 (CPG2) Inhibitor is a new CPG2 Inhibitor with antitumor activity.

Synonyms	Carboxypeptidase G2 Inhibitor, CPG2 Inhibitor
Molecular Weight	313.33
Formula	C13H15NO6S
CAS No.	192203-60-4

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 2 years

Solubility Information

H2O: 1.3 mg/mL (4.1 mM), Need ultrasonic

( < 1 mg/ml refers to the product slightly soluble or insoluble )

References and Literature

1. Khan, Tariq H.; Eno-Amooquaye, Ebun A.; Searle, Frances et al. Novel Inhibitors of Carboxypeptidase G2 (CPG2): Potential Use in Antibody-Directed Enzyme Prodrug Therapy. Journal of Medicinal Chemistry (1999), 42(6), 951-956. 2. Friedlos F, Lehouritis P, Ogilvie L et al. Attenuated Salmonella targets prodrug activating enzyme carboxypeptidase G2 to mouse melanoma and human breast and colon carcinomas for effective suicide gene therapy. Clin Cancer Res. 2008 Jul 1;14(13):4259-66. 3. Schepelmann S, Ogilvie LM, Hedley D et al. Suicide gene therapy of human colon carcinoma xenografts using an armed oncolytic adenovirus expressing carboxypeptidase G2. Cancer Res. 2007 May 15;67(10):4949-55. 4. Schepelmann S, Hallenbeck P, Ogilvie LM et al. Systemic gene-directed enzyme prodrug therapy of hepatocellular carcinoma using a targeted adenovirus armed with carboxypeptidase G2. Cancer Res. 2005 Jun 15;65(12):5003-8.

Related compound libraries

This product is contained In the following compound libraries：

Anti-Cancer Compound Library Bioactive Compounds Library Max Bioactive Compound Library

Related Products

Related compounds with same targets

CeMMEC1 2-PMPA 2-Benzylsuccinic acid CPA inhibitor CeMMEC13 BAY-299

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Method for preparing DMSO master liquid: mg drug pre-dissolved in μL DMSO (Master liquid concentration mg/mL)，Please contact us first if the concentration exceeds the DMSO solubility of the batch of drug.

Method for preparing in vivo formulation：Take μL DMSO master liquid, next add μL PEG300， mix and clarify, next add μL Tween 80，mix and clarify, next add μL ddH₂O, mix and clarify.

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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

Carboxypeptidase G2 (CPG2) Inhibitor 192203-60-4 Proteases/Proteasome Carboxypeptidase Carboxypeptidase G2 Inhibitor CPG2 Inhibitor inhibitor inhibit

Products are chemical reagents for research use only and are not intended for human use. We do not sell to patients.