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CCR1 antagonist 8

Catalog No. T14899 CAS 1295298-26-8

<a href="/target/CCR" style="display: inline; color: #c13a36">CCR</a>1 antagonist 8, a third azaindazole series compound, is a <a href="/target/CCR" style="display: inline; color: #c13a36">CCR</a>1 antagonist (IC50: 1.8 nM in Ca2+ flux assay).

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CCR1 antagonist 8, CAS 1295298-26-8

Pack Size	Availability	Price/USD
5 mg	14-16 weeks	$ 1,470.00
50 mg	14-16 weeks	$ 2,980.00
100 mg	14-16 weeks	$ 4,000.00

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Purity: 98%

Biological Description

Chemical Properties

Storage & Solubility Information

Description	CCR1 antagonist 8, a third azaindazole series compound, is a CCR1 antagonist (IC50: 1.8 nM in Ca2+ flux assay).
Targets&IC50	CCR1:1.8 nM （in Ca2+ flux assay)

Molecular Weight	451.47
Formula	C22H18FN5O3S
CAS No.	1295298-26-8

Storage

Powder: -20°C for 3 years

In solvent: -80°C for 2 years

Solubility Information

( < 1 mg/ml refers to the product slightly soluble or insoluble )

References and Literature

1. Harcken C, et al. Identification of novel azaindazole CCR1 antagonist clinical candidates. Bioorg Med Chem Lett. 2019 Feb 1;29(3):441-448.

Related Products

Related compounds with same targets

MLN-3897 BMS-817399 YM022 CCR1 antagonist 8 AZD2423 Aplaviroc ML218 GW 766994

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Keywords

CCR1 antagonist 8 1295298-26-8 Immunology/Inflammation Microbiology/Virology CCR CCR-1 antagonist 8 Inhibitor inhibitor inhibit

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