Powder: -20°C for 3 years
In solvent: -80°C for 2 years
BD1063 is a potent and selective sigma 1(σ1) receptor antagonist(Ki = 9 nM).
Description | BD1063 is a potent and selective sigma 1(σ1) receptor antagonist(Ki = 9 nM). |
In vivo | BD 1063 dose-dependently reduced ethanol self-administration in sP rats (3.3–11 mg/kg) and withdrawn, dependent Wistar rats (4–11 mg/kg) at doses that did not modify mean ethanol self-administration in non-dependent Wistar controls[1] |
Animal Research | Rats (controls, N=11;?dependent, N=9) were pretreated with BD-1063 (0, 4.4, 7 and 11 mg/kg of body weight, free base weights) using a within-subject Latin square design.?sP rats: Rats (N=9) were pretreated with BD-1063 (0, 3, 4.4, 7 and 11 mg/kg of body weight, free base basis) using a within-subject Latin square design[1]. |
Synonyms | BD1063 |
Molecular Weight | 346.12 |
Formula | C13H20Cl4N2 |
CAS No. | 206996-13-6 |
Powder: -20°C for 3 years
In solvent: -80°C for 2 years
H2O: 50 mg/mL (144.46 mM)
( < 1 mg/ml refers to the product slightly soluble or insoluble )
You can also refer to dose conversion for different animals. More
bottom
Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
BD1063 dhydrochloride 206996-13-6 G蛋白偶联受体 Sigma receptor Sigma Receptor Inhibitor inhibit BD1063 BD-1063 dhydrochloride inhibitor