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Azaline

Catalog No. T25129 CAS 134457-26-4

Synonyms: Azaline A

Azaline is a gonadorelin antagonist.

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Azaline, CAS 134457-26-4

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25 mg	Inquiry	$ 1,520.00

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Biological Description

Chemical Properties

Storage & Solubility Information

Description

Azaline is a gonadorelin antagonist.

Synonyms	Azaline A
Molecular Weight	1545.26
Formula	C74H106ClN23O12
CAS No.	134457-26-4

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

References and Literature

1. Ballantyne K, Anderson ST, Pyne M, Nicolson V, Mucci A, Lisle A, Johnston SD. Use of the gonadotrophin-releasing hormone antagonist azaline B to control the oestrous cycle in the koala (Phascolarctos cinereus). Reprod Fertil Dev. 2015 May 1. doi: 10.1071/RD14349. [Epub ahead of print] PubMed PMID: 25929179. 2. Chakraborty P, Roy SK. Effect of azaline B on follicular development and functions in the hamster. Mol Cell Endocrinol. 2015 Jan 15;400:1-9. doi: 10.1016/j.mce.2014.11.011. Epub 2014 Nov 24. PubMed PMID: 25462584; PubMed Central PMCID: PMC4274241. 3. Campen CA, Lai MT, Kraft P, Kirchner T, Phillips A, Hahn DW, Rivier J. Potent pituitary-gonadal axis suppression and extremely low anaphylactoid activity of a new gonadotropin releasing hormone (GnRH) receptor antagonist "azaline B". Biochem Pharmacol. 1995 May 11;49(9):1313-21. PubMed PMID: 7763313. 4. Rivier JE, Jiang G, Porter J, Hoeger CA, Craig AG, Corrigan A, Vale W, Rivier CL. Gonadotropin-releasing hormone antagonists: novel members of the azaline B family. J Med Chem. 1995 Jul 7;38(14):2649-62. PubMed PMID: 7629804.

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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

Azaline 134457-26-4 Azaline A inhibitor inhibit

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