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Alpidem

Catalog No. T26600 CAS 82626-01-5

Synonyms: Ananxyl

Alpidem (Ananxyl) is an anxiolytic drug from the imidazopyridine family. Alpidem does not produce sedative effects at normal doses, and is instead used specifically for the treatment of anxiety. Alpidem has nanomolar binding affinity for both the central benzodiaze

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Alpidem, CAS 82626-01-5

Pack Size	Availability	Price/USD
1 mg	In stock	$ 97.00
5 mg	In stock	$ 197.00
10 mg	In stock	$ 335.00
25 mg	In stock	$ 565.00
50 mg	In stock	$ 812.00
100 mg	In stock	$ 1,130.00
500 mg	In stock	$ 2,260.00
1 mL * 10 mM (in DMSO)	In stock	$ 375.00

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Purity: 100%

Purity: 99.49%

Biological Description

Chemical Properties

Storage & Solubility Information

Description

Synonyms	Ananxyl
Molecular Weight	404.33
Formula	C21H23Cl2N3O
CAS No.	82626-01-5

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

Solubility Information

DMSO: 30 mg/mL (74.2 mM)

References and Literature

1. Divya K Nair, et al. Synthesis of imidazopyridines from the Morita-Baylis-Hillman acetates of nitroalkenes and convenient access to Alpidem and Zolpidem. Org Lett. 2012 Sep 7;14(17):4580-3. 2. Natalia Chernyak, et al. General and efficient copper-catalyzed three-component coupling reaction towards imidazoheterocycles: one-pot synthesis of alpidem and zolpidem. Angew Chem Int Ed Engl. 2010 Apr 1;49(15):2743-6. 3. Andrea Cappelli, et al. Synthesis and structure-activity relationship studies in peripheral benzodiazepine receptor ligands related to alpidem. Bioorg Med Chem. 2008 Mar 15;16(6):3428-37. 4. Giuseppe Trapani, et al. Alpidem analogues containing a GABA or glycine moiety as new anticonvulsant agents. Eur J Pharm Sci. 2003 Mar;18(3-4):231-40.

Related compound libraries

This product is contained In the following compound libraries：

Membrane Protein-targeted Compound Library Anti-Neurodegenerative Disease Compound Library Drug-induced Liver Injury (DILI) Compound Library Human Metabolite Library Neurotransmitter Receptor Compound Library Bioactive Compounds Library Max Bioactive Compound Library Neuronal Signaling Compound Library Anti-Cancer Compound Library ReFRAME Related Library

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Method for preparing DMSO master liquid: mg drug pre-dissolved in μL DMSO (Master liquid concentration mg/mL)，Please contact us first if the concentration exceeds the DMSO solubility of the batch of drug.

Method for preparing in vivo formulation：Take μL DMSO master liquid, next add μL PEG300， mix and clarify, next add μL Tween 80，mix and clarify, next add μL ddH₂O, mix and clarify.

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What is the mass of compound required to make a 10 mM stock solution in 10 ml of water given that the molecular weight of the compound is 197.13 g/mol?
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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

Alpidem 82626-01-5 Membrane transporter/Ion channel Neuroscience GABA Receptor Ananxyl inhibit Gamma-aminobutyric acid Receptor Inhibitor γ-Aminobutyric acid Receptor inhibitor

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