Powder: -20°C for 3 years | In solvent: -80°C for 1 year
[(3S)-3-amino-4-(3-hexylanilino)-4-oxobutyl]phosphonic acid;hydrobromide is a S1P1 antagonist with Ki of 2.84 μM.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 195.00 | |
2 mg | In stock | $ 293.00 | |
5 mg | In stock | $ 447.00 | |
10 mg | In stock | $ 659.00 | |
25 mg | In stock | $ 987.00 | |
50 mg | In stock | $ 1,380.00 | |
100 mg | In stock | $ 1,890.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 498.00 |
Description | [(3S)-3-amino-4-(3-hexylanilino)-4-oxobutyl]phosphonic acid;hydrobromide is a S1P1 antagonist with Ki of 2.84 μM. |
In vitro | In a GTP-gSbindingassay, activation of hS1P1 receptors by physiological agonist S1P alone or in the presence of 10 μM [(3S)-3-amino-4-(3-hexylanilino)-4-oxobutyl]phosphonic acid;hydrobromide, the EC50 value was 0.8 nM or 50nM, respectively. |
Molecular Weight | 423.28 |
Formula | C16H28BrN2O4P |
CAS No. | 1246817-25-3 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 55 mg/mL (129.94 mM)
You can also refer to dose conversion for different animals. More
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W140 HBr 1246817-25-3 GPCR/G Protein S1P Receptor [(3S)3amino4(3hexylanilino)4oxobutyl]phosphonicacid;hydrobromide inhibitor inhibit