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(R)-(-)-α-Methylhistamine dihydrochloride

Catalog No. T24698 CAS 75614-89-0

Synonyms: HISTAMINE DIHYDROCHLORIDE R(-)-A-METHYL

R(-)-alpha-Methylhistamine 2HCl is an effective and selective agonist of the H3 histamine receptor.

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(R)-(-)-α-Methylhistamine dihydrochloride Chemical Structure

(R)-(-)-α-Methylhistamine dihydrochloride, CAS 75614-89-0

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Biological Description

Chemical Properties

Storage & Solubility Information

Description	R(-)-alpha-Methylhistamine 2HCl is an effective and selective agonist of the H3 histamine receptor.
Targets&IC50	H3 receptor:50.3 nM (Kd)

Synonyms	HISTAMINE DIHYDROCHLORIDE R(-)-A-METHYL
Molecular Weight	198.09
Formula	C6H13Cl2N3
CAS No.	75614-89-0

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

References and Literature

1. Lamberti C, Bartolini A, Ghelardini C, Malmberg-Aiello P. Investigation into the role of histamine receptors in rodent antinociception. Pharmacol Biochem Behav. 1996 Mar;53(3):567-74. PubMed PMID: 8866956. 2. Malmberg-Aiello P, Lamberti C, Ghelardini C, Giotti A, Bartolini A. Role of histamine in rodent antinociception. Br J Pharmacol. 1994 Apr;111(4):1269-79. PubMed PMID: 8032614; PubMed Central PMCID: PMC1910136.

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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

(R)-(-)-α-Methylhistamine dihydrochloride 75614-89-0 HISTAMINE DIHYDROCHLORIDE RA-METHYL alpha-Methylhistamine a-Methylhistamine alpha-Methylhistamine Dihydrochloride HISTAMINE DIHYDROCHLORIDE R(-)-A-METHYL α-Methylhistamine Dihydrochloride (R)()αMethylhistamine dihydrochloride a-Methylhistamine Dihydrochloride α-Methylhistamine (R) ( ) α Methylhistamine dihydrochloride inhibitor inhibit

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