Powder: -20°C for 3 years | In solvent: -80°C for 1 year
(±)-J-113397 is a potent and selective non-peptidyl ORL1 receptor antagonist (K(i): cloned human ORL1=1.8 nM). J-113397 inhibited nociceptin/orphanin FQ-stimulated GTPγS binding to CHO cells expressing ORL1 with an IC 50 value of 5.3 nM. J-113397 can be used for researching the physiological roles of nociceptin/orphanin FQ [1].
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
25 mg | 10-14 weeks | $ 931.00 | |
50 mg | 10-14 weeks | $ 1,210.00 | |
100 mg | 10-14 weeks | $ 1,830.00 |
Description | (±)-J-113397 is a potent and selective non-peptidyl ORL1 receptor antagonist (K(i): cloned human ORL1=1.8 nM). J-113397 inhibited nociceptin/orphanin FQ-stimulated GTPγS binding to CHO cells expressing ORL1 with an IC 50 value of 5.3 nM. J-113397 can be used for researching the physiological roles of nociceptin/orphanin FQ [1]. |
Molecular Weight | 399.57 |
Formula | C24H37N3O2 |
CAS No. | 217461-40-0 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
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(±)-J 113397 217461-40-0 J 113397 (±)J 113397 (±) J 113397 J-113397 J113397 inhibitor inhibit