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GSK-5959  
Catalog No. T1972    CAS 901245-65-6
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5mg
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85.00
10mg
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136.00
25mg
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327.00
50mg
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638.00
1g
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0.00
5g
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0.00
10 mM * 1 mL (in DMSO)
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94.00
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Documents and Quality Management
Purity:98.65% COA Datasheet HNMR HPLC
Biological Activity:

Product Description:

GSK-5959 is an effective, specific and cell permeable BRPF1 bromodomain inhibitor (IC50: ~80 nM). The selectivity of GSK-5959 for BRPF1 is >100-fold over a panel of 35 other bromodomains, including BRPF2/3 and BET family bromodomains.

Target:
BRPF1;
Research Area:
Other
Chemical Information:
Molecular Weight 394.47
Formula C22H26N4O3
CAS Number 901245-65-6
Solubility DMSO:10 mM
Storage 3 years -20°C powder;
2 years -80°C in solvent;
Remark For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ℃ for several month.
Technical Support

Answers to questions you may have can be found in the inhibitor handling instructions. Topics include how to prepare stock solutions, how to store Products, and issues that need special attention for cell-based assays and animal experiments.

Related Compound Libraries
This product is contained In the following compound libraries:
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Reference

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