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Entinostat (MS-275)  
Catalog No. T6233    CAS 209783-80-2
Pack Size
Availability
Price/USD
Quantity
5mg
In Stock
32.00
25mg
In Stock
57.00
50mg
In Stock
79.00
100mg
In Stock
109.00
10mM * 1mL (in DMSO)
In Stock
48.00
10mg
In Stock
45.00
Bulk Size: Please Quote for Discount
Documents and Quality Management
Purity:98.00% COA Datasheet HNMR HPLC MSDS
Biological Activity:

Product Description:

Entinostat (MS-275) strongly inhibits HDAC1 and HDAC3 with IC50 of 0.51 μM and 1.7 μM, compared with HDACs 4, 6, 8, and 10. Phase 3.

Target:
HDAC3; HDAC1;
Research Area:
Cancer
Chemical Information:
Molecular Weight 376.41
Formula C21H20N4O3
CAS Number 209783-80-2
Solubility DMSO: 75mg/ml(199.25 mM);Water: <1mg/ml;Ethanol: <1mg/ml
Storage 3 years -20°C powder;
2 years -80°C in solvent;
Remark For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ℃ for several month.
Technical Support

Answers to questions you may have can be found in the inhibitor handling instructions. Topics include how to prepare stock solutions, how to store Products, and issues that need special attention for cell-based assays and animal experiments.

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Reference

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