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Aurora-Kinase
Cat.No. Product Name Information Area
T6936 PF-03814735 PF-03814735 is a novel, potent and reversible inhibitor of Aurora A/B with IC50of 0.8... Others
T6785 BI-847325 BI-847325 is a selective dual inhibitor of MEK and aurora kinases (AK) with IC50 valu... Others
T6767 Aurora A Inhibitor I Aurora A Inhibitor I is a novel, potent, and selective inhibitor of Aurora A with IC5... Others
T6458 CYC116 CYC116 is a potent inhibitor of Aurora A/B with Ki of 8.0 nM/9.2 nM, is less potent t... Cancer
T6380 AMG-900 AMG 900 is a potent and highly selective pan-Aurora kinases inhibitor for Aurora A/B/... Cancer
T6435 CCT129202 CCT129202 is an ATP-competitive pan-Aurora inhibitor for Aurora A, Aurora B and Auror... Cancer
T6077 ZM 447439 ZM 447439 is a selective and ATP-competitive inhibitor for Aurora A and Aurora B with... Cancer
T6068 MK-5108 (VX-689) MK-5108 is a highly potent and specific Aurora-A kinase inhibitor with an IC50 value ... Cancer
T3068 AT9283 AT9283 is an effective multi-targeted inhibitor of JAK2(IC50=1.2 nM) and JAK3(IC50=1... Cancer
T2709 TAK901 TAK-901 has been used in trials studying the treatment of Lymphoma, Myelofibrosis, Mu... Cancer
T2699 BMS-777607 BMS-777607 is a Met-related inhibitor for c-Met/Axl/Ron/Tyro3 (IC50: 3.9/1.1/1.8/4.3 ... Endocrine system
T2620 G-749 G-749, a new-type FLT3 inhibitor, exhibits effective and sustained inhibition of the ... Cardiovascular System
T2617 SNS-314 Mesylate SNS-314 Mesylate is an effective and specific Aurora A/B/C inhibitor (IC50: 9/31/3 nM... Cancer
T2611 CCT 137690 CCT 137690 is a highly specific and oral-available aurora kinase inhibitor, for auro... Cancer
T2602 AZD1152-HQPA Barasertib (AZD1152-HQPA) is a highly selective Aurora B inhibitor (IC50: 0.37 nM) i... Cancer
T2509 Tozasertib VX-680 (Tozasertib, MK-0457) is a pan-Aurora inhibitor, mostly against Aurora A (Kiap... Cancer
T2471 MK8745 MK-8745 is a potent and selective Aurora A inhibitor. Cancer
T2358 ENMD-2076 ENMD-2076, a multi-targeted kinase inhibitor, has specific activity against Aurora A,... Cancer
T2349 BMS-754807 Dual IGF-1R/InsR Inhibitor BMS-754807 is an oral small molecule inhibitor of insulin-... Cancer
T2241 Alisertib Alisertib (MLN8237) is a specific Aurora A inhibitor (IC50: 1.2 nM). The selectivity ... Cancer
T2094 Danusertib Danusertib is a small-molecule 3-aminopyrazole derivative with potential antineoplast... Cancer
T1825 Reversine Reversine, a small synthetic purine analogue (2,6-disubstituted purine), is a potent ... Other
T6338 PHA-680632 PHA-680632 is potent inhibitor of Aurora A, Aurora B and Aurora C with IC50 of 27 nM,... Cancer
T6315 MLN8054 MLN8054 is a potent and selective Aurora A kinase inhibitor with an IC50 of 4 nM. Cancer
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