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GR 94800 acetate

Name: GR 94800 acetate
Brand: TargetMol
SKU: T22811L
Price: 382 USD
Availability: InStock
Rating: 5 (10 reviews)

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Catalog No. T22811L

Alias GR 94800 acetate (141636-65-9 free base)

GR 94800 acetate is a potent and selective neurokinin 2(NK-2) antagonist.

GR 94800 acetate

🥰Excellent

Purity: 97.86%

Catalog No. T22811LAlias GR 94800 acetate (141636-65-9 free base)

GR 94800 acetate is a potent and selective neurokinin 2(NK-2) antagonist.

Pack Size	Price	USA Warehouse	Global Warehouse
1 mg	$382	-	In Stock
2 mg	$542	-	In Stock
5 mg	$816	-	In Stock
10 mg	$1,090	-	In Stock
25 mg	$1,630	-	In Stock
50 mg	$2,200	-	In Stock
100 mg	$2,970	-	In Stock

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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]

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Purity:97.86%

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COA HPLC MS

Product Introduction

Bioactivity

Description	GR 94800 acetate is a potent and selective neurokinin 2(NK-2) antagonist.
Targets&IC50	NK2:9.6(pKb), NK3:6.0(pKb), NK1:6.4(pKb)
In vitro	GR 94800 displayed high affinity (pIC50 8.4-9.5) with no significant difference in potency between these four tissues from the rat fundus, colon, bladder and vas deferens[3].
Synonyms	GR 94800 acetate (141636-65-9 free base)

Chemical Properties

Molecular Weight	964.12
Formula	C₅₁H₆₅N₉O₁₀
Smiles	CCCC[C@@H](C(N)=O)NC([C@H](CCC1)N1C([C@@H](CCC1)N1C([C@H](Cc1ccccc1)NC([C@@H](Cc1c[nH]c2c1cccc2)NC([C@H](C)NC([C@H](C)NC(c1ccccc1)=O)=O)=O)=O)=O)=O)=O.CC(O)=O
Color	White
Appearance	Solid
Sequence	Bz-Ala-Ala-Trp-Phe-Pro-Pro-Nle
Sequence Short	AAWFPPX

Storage & Solubility Information

Storage

keep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

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