Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Sematilide is a blocker of selective IKr channel.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
25 mg | 6-8 weeks | $ 1,520.00 | |
50 mg | 6-8 weeks | $ 1,980.00 | |
100 mg | 6-8 weeks | $ 2,500.00 |
Description | Sematilide is a blocker of selective IKr channel. |
Targets&IC50 | K+ current:25 μM |
In vitro | Sematilide(10, 30, 100 and 300 μM) causes a concentration-dependent inhibition of the delayed rectifier K+ current with IC50 of 25 μM[1]. |
In vivo | Sematilide in 0.3-1.0 mg/kg(intravenously i.v.) is effective in a canine model of arrhythmia[2]. |
Synonyms | CK-1752 |
Molecular Weight | 313.42 |
Formula | C14H23N3O3S |
CAS No. | 101526-83-4 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
You can also refer to dose conversion for different animals. More
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Sematilide 101526-83-4 Others CK-1752 CK 1752 CK1752 inhibitor inhibit