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Protease-Activated Receptor-2, amide

Catalog No. T7513   CAS 190383-13-2
Synonyms: SLIGKV-NH2

Protease-Activated Receptor-2, amide (SLIGKV-NH2) is an agonist of PAR2 (IC50 : 10.4 M)

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Protease-Activated Receptor-2, amide Chemical Structure
Protease-Activated Receptor-2, amide, CAS 190383-13-2
Pack Size Availability Price/USD Quantity
2 mg In stock $ 48.00
5 mg In stock $ 70.00
10 mg In stock $ 118.00
25 mg In stock $ 201.00
50 mg In stock $ 302.00
100 mg In stock $ 453.00
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Purity: 100%
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Biological Description
Chemical Properties
Storage & Solubility Information
Description Protease-Activated Receptor-2, amide (SLIGKV-NH2) is an agonist of PAR2 (IC50 : 10.4 M)
Targets&IC50 PAR2:10.4 M
Synonyms SLIGKV-NH2
Molecular Weight 614.78
Formula C28H54N8O7
CAS No. 190383-13-2

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

Solubility Information

H2O: 33.33 mg/mL (54.21 mM), sonification is recommended.

TargetMolReferences and Literature

1. Kanke T , Ishiwata H , Kabeya M , et al. Binding of a highly potent protease-activated receptor-2 (PAR2) activating peptide, [~3H]2-furoyl-LIGRL-NH_2, to human PAR2[J]. British Journal of Pharmacology, 2005, 145(2):p.255-263.

Related compound libraries

This product is contained In the following compound libraries:
Peptide Compound Library NO PAINS Compound Library

Related Products

Related compounds with same targets
TFLLR-NH2 Protease-Activated Receptor-1, PAR-1 Agonist acetate Vorapaxar TRAP-6 amide acetate PAR-4 Agonist Peptide, amide TFA AC-264613 Thrombin Receptor Activator for Peptide 5 (TRAP-5) 2-Furoyl-LIGRLO-amide TFA(729589-58-6 free base)

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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

Protease-Activated Receptor-2, amide 190383-13-2 GPCR/G Protein Protease-activated Receptor ProteaseActivated Receptor2, amide Protease Activated Receptor (PAR) Inhibitor Thrombin receptors inhibit Protease Activated Receptor 2, amide SLIGKV-NH2 Protease-Activated Receptor-2, Amide inhibitor

 

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