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GPCR/G Protein Protease-activated Receptor Protease-Activated Receptor-2, amide

Protease-Activated Receptor-2, amide

Catalog No. T7513   CAS 190383-13-2

Protease-Activated Receptor-2, amide is an agonist of PAR2 (IC50 : 10.4 M)

Protease-Activated Receptor-2, amide, CAS 190383-13-2
Pack Size Availability Price/USD Quantity
2 mg In stock 54.00
5 mg In stock 78.00
10 mg In stock 132.00
25 mg In stock 224.00
50 mg In stock 336.00
100 mg In stock 504.00
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Purity 100.00%
Biological Description
Chemical Properties
Storage & Solubility Information
Description Protease-Activated Receptor-2, amide is an agonist of PAR2 (IC50 : 10.4 M)
Targets&IC50 PAR2 : ic50 10.4 M,  
Molecular Weight 614.78
Formula C28H54N8O7
CAS No. 190383-13-2

Storage

0-4℃ for short term (days to weeks), or -20℃ for long term (months).

Solubility Information

H2O: 33.33 mg/mL (54.21 mM), Need ultrasonic

( < 1 mg/ml refers to the product slightly soluble or insoluble )

Citations

References and Literature
1. Kanke T, et al. Binding of a highly potent protease-activated receptor-2 (PAR2) activating peptide, [3H]2-furoyl-LIGRL-NH2, to human PAR2. Br J Pharmacol. 2005 May;145(2):255-63. 1. Kanke T , Ishiwata H , Kabeya M , et al. Binding of a highly potent protease-activated receptor-2 (PAR2) activating peptide, [~3H]2-furoyl-LIGRL-NH_2, to human PAR2[J]. British Journal of Pharmacology, 2005, 145(2):p.255-263.

Related Products

Related compounds with same targets
TFLLR-NH2 2TFA(197794-83-5(free base)) Thrombin Receptor Activator for Peptide AZ3451 Thrombin Receptor Activator for Peptide Protease-Activated Receptor-4 diTFA(245443-52-1(free base)) PAR-4 Agonist Peptide, amide TFA 2-Furoyl-LIGRLO-amide TFA(729589-58-6 free base) AC264613

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