Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Divaplon is a GABA receptor agonist (IC50: 0.056 µM) that displays non-sedating anxiolytic behavioral characteristics in a rat model of anxiety.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 146.00 | |
5 mg | In stock | $ 350.00 | |
10 mg | In stock | $ 530.00 | |
25 mg | In stock | $ 859.00 | |
50 mg | In stock | $ 1,180.00 | |
100 mg | In stock | $ 1,590.00 | |
500 mg | In stock | $ 3,190.00 |
Description | Divaplon is a GABA receptor agonist (IC50: 0.056 µM) that displays non-sedating anxiolytic behavioral characteristics in a rat model of anxiety. |
In vivo | Divaplon (1-60 mg/kg; injection; mice) clearly produced effects on the acquisition of conditioned fear. As the drug has been shown to produce anticonvulsant and anxiolytic-like effects without sedation or depression of motor activity. The results show that BZ (omega) receptor partial agonists without apparent sedative actions can disrupt fear learning, indicating that the effects of this class of drugs on passive avoidance learning can be dissociated from sedation.[4] |
Synonyms | RU-32698, RU32698, RU 32698 |
Molecular Weight | 295.34 |
Formula | C17H17N3O2 |
CAS No. | 90808-12-1 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 50 mg/mL (169.3 mM)
You can also refer to dose conversion for different animals. More
bottom
Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
Divaplon 90808-12-1 Membrane transporter/Ion channel Neuroscience GABA Receptor RU-32698 RU32698 RU 32698 inhibitor inhibit