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CCR1 antagonist 6

Catalog No. T10708 CAS 2436773-01-0

<a href="/target/CCR" style="display: inline; color: #c13a36">CCR</a>1 antagonist 6 (compound 16q) is an antagonist of chemokine receptor 1 (<a href="/target/CCR" style="display: inline; color: #c13a36">CCR</a>1) with an IC 50 of 3 nM [1].

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CCR1 antagonist 6, CAS 2436773-01-0

Pack Size	Availability	Price/USD
5 mg	Synthesizing, 8-12 weeks	$ 970.00
50 mg	Synthesizing, 8-12 weeks	$ 1,980.00
100 mg	Synthesizing, 8-12 weeks	$ 2,500.00

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Purity: 98%

Biological Description

Chemical Properties

Storage & Solubility Information

Description	CCR1 antagonist 6 (compound 16q) is an antagonist of chemokine receptor 1 (CCR1) with an IC 50 of 3 nM [1].
Targets&IC50	CCR1:3 nM

Molecular Weight	446.95
Formula	C21H23ClN4O3S
CAS No.	2436773-01-0

Storage

Powder: -20°C for 3 years

In solvent: -80°C for 2 years

Solubility Information

( < 1 mg/ml refers to the product slightly soluble or insoluble )

References and Literature

1. Harcken C, et al. Discovery and optimization of pyrazole amides as antagonists of CCR1. Bioorg Med Chem Lett. 2019 Feb 1;29(3):435-440.

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Keywords

CCR1 antagonist 6 2436773-01-0 Immunology/Inflammation Microbiology/Virology CCR CCR-1 antagonist 6 Inhibitor inhibitor inhibit

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