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P2X4 antagonist-1

Name: P2X4 antagonist-1
Brand: TargetMol
SKU: T87086
Price: 48 USD
Availability: InStock
Rating: 5 (10 reviews)

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Catalog No. T87086Cas No. 2055601-42-6

P2X4 antagonist-1 is a potent P2X4 receptor antagonist used in the study of neurological, cardiovascular, and immune system diseases.

P2X4 antagonist-1

🥰Excellent

Purity: 99.9%

Catalog No. T87086Cas No. 2055601-42-6

P2X4 antagonist-1 is a potent P2X4 receptor antagonist used in the study of neurological, cardiovascular, and immune system diseases.

Pack Size	Price	Availability
1 mg	$48	In Stock
5 mg	$113	In Stock
10 mg	$179	In Stock
25 mg	$355	In Stock
50 mg	$569	In Stock
100 mg	$892	In Stock
200 mg	$1,220	In Stock

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Batch Information

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Purity:99.9%

Resource Download

COA HNMR HPLC

Product Introduction

Bioactivity

Description	P2X4 antagonist-1 is a potent P2X4 receptor antagonist used in the study of neurological, cardiovascular, and immune system diseases.
Targets&IC50	P2X4 receptor:15 nM
In vitro	P2X4 antagonist-1 (Compound 24) is an antagonist targeting the P2X4 receptor with an IC50 of 15 nM. [1]

Chemical Properties

Molecular Weight	485.77
Formula	C₂₀H₁₅Cl₃N₂O₄S
Cas No.	2055601-42-6
Smiles	O=C(NC1=CC=C(OC=2C=CC=C(Cl)C2)C(=C1)S(=O)(=O)N)CC=3C(Cl)=CC=CC3Cl
Color	White
Appearance	Solid

Storage & Solubility Information

Storage

store at low temperature | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.

Solubility Information

DMSO: 80 mg/mL (164.69 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	2.0586 mL	10.2929 mL	20.5859 mL	102.9294 mL
5 mM	0.4117 mL	2.0586 mL	4.1172 mL	20.5859 mL
10 mM	0.2059 mL	1.0293 mL	2.0586 mL	10.2929 mL
20 mM	0.1029 mL	0.5146 mL	1.0293 mL	5.1465 mL
50 mM	0.0412 mL	0.2059 mL	0.4117 mL	2.0586 mL
100 mM	0.0206 mL	0.1029 mL	0.2059 mL	1.0293 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc