OPC-14523 free base

Name: OPC-14523 free base
Brand: TargetMol
SKU: T28256
Rating: 4.5 (1 reviews)

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Catalog No. T28256Cas No. 145969-30-8

Alias VPI-013, VPI013, VPI 013, OPC-14523, OPC14523, OPC 14523

OPC-14523, a 5-HT1A receptor agonist, is used potentially for the treatment of depression and neuropathic pain.

OPC-14523 free base

😃Good

Catalog No. T28256Alias VPI-013, VPI013, VPI 013, OPC-14523, OPC14523, OPC 14523Cas No. 145969-30-8

OPC-14523, a 5-HT1A receptor agonist, is used potentially for the treatment of depression and neuropathic pain.

Pack Size	Price	Availability
25 mg	$1,520	6-8 weeks
50 mg	$1,980	6-8 weeks
100 mg	$2,500	6-8 weeks

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This molecule is a custom-made product. TargetMol has an excellent synthesis team with the experience and capability to provide you with cost-effective products. However, due to objective factors, there is a small probability that the synthesis may not be successful during the R&D process. We appreciate your understanding. If you have any questions, please feel free to contact us. We are committed to serving you wholeheartedly.

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Product Introduction

Bioactivity

Description	OPC-14523, a 5-HT1A receptor agonist, is used potentially for the treatment of depression and neuropathic pain.
Targets&IC50	5-HT1A receptor:2.3 nM (IC50), σ1:47 nM (IC50), σ2:56 nM (IC50)
Synonyms	VPI-013, VPI013, VPI 013, OPC-14523, OPC14523, OPC 14523

Chemical Properties

Molecular Weight	413.94
Formula	C₂₃H₂₈ClN₃O₂
Cas No.	145969-30-8
Relative Density.	no data available

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

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DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

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Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

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