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BD 1008 dihydrobromide

🥰Excellent
Catalog No. T21788Cas No. 138356-09-9

BD 1008 dihydrobromide is a selective antagonist of the sigma 1 (σ1) receptor (Ki = 2 nM). BD 1008 dihydrobromide have high affinity for sigma1 receptors, moderate affinity for sigma2 receptors.

BD 1008 dihydrobromide
Other Forms of BD 1008 dihydrobromide:
BD 1008 Free BaseT70809138356-08-8
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BD 1008 dihydrobromide

🥰Excellent
Purity: 97.81%
Catalog No. T21788Cas No. 138356-09-9
BD 1008 dihydrobromide is a selective antagonist of the sigma 1 (σ1) receptor (Ki = 2 nM). BD 1008 dihydrobromide have high affinity for sigma1 receptors, moderate affinity for sigma2 receptors.
Pack SizePriceUSA WarehouseGlobal WarehouseQuantity
2 mg$35In StockIn Stock
5 mg$56In StockIn Stock
10 mg$98In StockIn Stock
25 mg$239In StockIn Stock
50 mg$373In StockIn Stock
100 mg$531-In Stock
1 mL x 10 mM (in DMSO)$73In StockIn Stock
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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.
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Batch Information

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Purity:97.81%
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Product Introduction

Bioactivity
Description
BD 1008 dihydrobromide is a selective antagonist of the sigma 1 (σ1) receptor (Ki = 2 nM). BD 1008 dihydrobromide have high affinity for sigma1 receptors, moderate affinity for sigma2 receptors.
Targets&IC50
σ1 receptor:2 nM(Ki)
Chemical Properties
Molecular Weight463.08
FormulaC15H24Br2Cl2N2
Cas No.138356-09-9
Smiles[H]Br.[H]Br.CN(CCC1=CC=C(Cl)C(Cl)=C1)CCN2CCCC2
Relative Density.no data available
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
Solubility Information
DMSO: 32.5 mg/mL (70.18 mM), Sonication is recommended.
Solution Preparation Table
DMSO
1mg5mg10mg50mg
1 mM2.1595 mL10.7973 mL21.5945 mL107.9727 mL
5 mM0.4319 mL2.1595 mL4.3189 mL21.5945 mL
10 mM0.2159 mL1.0797 mL2.1595 mL10.7973 mL
20 mM0.1080 mL0.5399 mL1.0797 mL5.3986 mL
50 mM0.0432 mL0.2159 mL0.4319 mL2.1595 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
TargetMol | Animal experimentsFor example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH2O. So your working solution concentration is 2 mg/mL。
Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH2OTargetMol | reagent mix well and clarify
For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.
1 Enter information below:
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2 Enter the in vivo formulation:
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%
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Dose Conversion

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc

Keywords

σ1SigmareceptorSigma receptorBD-1008 DihydrobromideBD1008 DihydrobromideBD-1008BD1008BD 1008 dihydrobromideBD 1008 DihydrobromideBD 1008
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