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GPCR/G Protein OX Receptor Orexin 2 Receptor Agonist

Orexin 2 Receptor Agonist

Catalog No. T3177   CAS 1796565-52-0
Synonyms: OX2R

Orexin 2 Receptor Agonist is an effective (EC50: 23 nM) and OX2R-selective (OX1R/OX2R EC50 ratio: 70) agonist.

Orexin 2 Receptor Agonist, CAS 1796565-52-0
Pack Size Availability Price/USD Quantity
1 mg In stock 50.00
2 mg In stock 90.00
5 mg In stock 135.00
10 mg In stock 193.00
25 mg In stock 370.00
50 mg In stock 650.00
1 mL * 10 mM (in DMSO) In stock 193.00
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Biological Description
Chemical Properties
Storage & Solubility Information
Description Orexin 2 Receptor Agonist is an effective (EC50: 23 nM) and OX2R-selective (OX1R/OX2R EC50 ratio: 70) agonist.
Targets&IC50 O2XR : ic50 23nM,  
Synonyms OX2R
Purity 99.43%
Molecular Weight 586.7
Formula C32H34N4O5S
CAS No. 1796565-52-0

Storage

0-4℃ for short term (days to weeks), or -20℃ for long term (months).

Solubility Information

DMSO: 32 mg/mL

( < 1 mg/ml refers to the product slightly soluble or insoluble )

Citations

References and Literature
1. Nagahara T, et al. J Med Chem. 2015 Oct 22;58(20):7931-7. 2. Nagahara T, et al. Design and Synthesis of Non-Peptide, Selective Orexin Receptor 2 Agonists. J Med Chem. 2015 Oct 22;58(20):7931-7.

Related compound libraries

This product is contained In the following compound libraries:
Bioactive Compound Library Inhibitor Library Neuronal Signaling Compound Library GPCR Compound Library

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