Powder: -20°C for 3 years
In solvent: -80°C for 2 years
Highly potent melanocortin MC4 receptor antagonist (Ki values are 0.29, 18.6, 5.45 and 3.29 nM for cloned human MC4, MC1, MC3 and MC5 receptors respectively). Increases food intake, and blocks α-MSH- and MTII-induced hypotension and bradycardia in rats, following central administration in vivo.
Description | Highly potent melanocortin MC4 receptor antagonist (Ki values are 0.29, 18.6, 5.45 and 3.29 nM for cloned human MC4, MC1, MC3 and MC5 receptors respectively). Increases food intake, and blocks α-MSH- and MTII-induced hypotension and bradycardia in rats, following central administration in vivo. |
Synonyms | HS 024 |
Molecular Weight | 1266.5 |
Formula | C58H79N19O10S2 |
CAS No. | 212370-59-7 |
Powder: -20°C for 3 years
In solvent: -80°C for 2 years
H2O: 0.50 mg/mL
( < 1 mg/ml refers to the product slightly soluble or insoluble )
You can also refer to dose conversion for different animals. More
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HS024 212370-59-7 GPCR/G Protein Neuroscience Melanocortin Receptor selective melanocortin intake Inhibitor MC Receptor HS-024 food HS 024 inhibit inhibitor