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Endothelial lipase inhibitor-1

Catalog No. T11199 CAS 1466427-02-0

Endothelial <a href="/target/Lipase" style="display: inline; color: #c13a36">Lipase</a> inhibitor-1 is a potent endothelial <a href="/target/Lipase" style="display: inline; color: #c13a36">Lipase</a> inhibitor with an IC50 of 49 nM.

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Endothelial lipase inhibitor-1, CAS 1466427-02-0

Pack Size	Availability	Price/USD
1 mg	In stock	$ 354.00
5 mg	In stock	$ 678.00
10 mg	In stock	$ 1,128.00
25 mg	In stock	$ 1,965.00
50 mg	In stock	$ 2,944.00
100 mg	In stock	$ 4,418.00
1 mL * 10 mM (in DMSO)	In stock	$ 833.00

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Purity: 97.38%

Biological Description

Chemical Properties

Storage & Solubility Information

Description	Endothelial lipase inhibitor-1 is a potent endothelial lipase inhibitor with an IC50 of 49 nM.
Targets&IC50	endothelial lipase:49 nM

Molecular Weight	406.43
Formula	C22H22N4O4
CAS No.	1466427-02-0

Storage

Powder: -20°C for 3 years

In solvent: -80°C for 2 years

Solubility Information

DMSO: 20 mg/mL (49.2 mM), Need ultrasonic

( < 1 mg/ml refers to the product slightly soluble or insoluble )

References and Literature

1. Hu CH, et al. Discovery and synthesis of tetrahydropyrimidinedione-4-carboxamides as endothelial lipase inhibitors. Bioorg Med Chem Lett. 2018 Dec 15;28(23-24):3721-3725.

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Keywords

Endothelial lipase inhibitor-1 1466427-02-0 Metabolism Lipase Endothelial lipase inhibitor1 Endothelial lipase inhibitor 1 Inhibitor inhibitor inhibit

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