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Eg5 Inhibitor V, trans-24

Catalog No. T11155 CAS 869304-55-2

Eg5 Inhibitor V, trans-24 is a specific and potent Eg5 inhibitor that can be used in cancer research with an IC50 value of 0.65 uM.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

Eg5 Inhibitor V, trans-24, CAS 869304-55-2

Pack Size	Availability	Price/USD
1 mg	In stock	$ 155.00
2 mg	In stock	$ 233.00
5 mg	In stock	$ 358.00
10 mg	In stock	$ 536.00
25 mg	In stock	$ 867.00
50 mg	In stock	$ 1,190.00
100 mg	In stock	$ 1,590.00
1 mL * 10 mM (in DMSO)	In stock	$ 398.00

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Purity: 97.45%

Biological Description

Chemical Properties

Storage & Solubility Information

Description	Eg5 Inhibitor V, trans-24 is a specific and potent Eg5 inhibitor that can be used in cancer research with an IC50 value of 0.65 uM.
Targets&IC50	Eg5:0.65 μM
In vitro	Trans-24 is a potent EG5-specific inhibitor with an IC50 conversion rate of 0.65 M and can be used in cancer research[1].

Molecular Weight	423.46
Formula	C26H21N3O3
CAS No.	869304-55-2

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 2 years

Solubility Information

DMSO: 45 mg/mL (106.27 mM)

( < 1 mg/ml refers to the product slightly soluble or insoluble )

References and Literature

1. Sunder-Plassmann N, et al. Synthesis and biological evaluation of new tetrahydro-beta-carbolines as inhibitors of the mitotic kinesin Eg5. Bioorg Med Chem. 2005 Nov 15;13(22):6094-111.

Related compound libraries

This product is contained In the following compound libraries：

Bioactive Compound Library Inhibitor Library Anti-Cancer Compound Library Cytoskeletal Signaling Pathway Compound Library Bioactive Compounds Library Max

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Method for preparing DMSO master liquid: mg drug pre-dissolved in μL DMSO (Master liquid concentration mg/mL)，Please contact us first if the concentration exceeds the DMSO solubility of the batch of drug.

Method for preparing in vivo formulation：Take μL DMSO master liquid, next add μL PEG300， mix and clarify, next add μL Tween 80，mix and clarify, next add μL ddH₂O, mix and clarify.

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Be sure to add the solvent(s) in order. Physical methods such as vortex, ultrasound or hot water bath can be used to aid dissolving.

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

Eg5 Inhibitor V, trans-24 869304-55-2 Cytoskeletal Signaling Kinesin Eg5 Inhibitor V, trans 24 Eg-5 Inhibitor V, trans-24 Eg5 Inhibitor V, trans24 inhibitor inhibit

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