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TargetMol | Compound Library

Anti-Cancer Active Compound Library

Catalog No. L2160

During the past decades, we have witnessed many landmark discoveries and successes in cancer research and therapy, however, cancer is still a major health problem for human beings, and it often physically and emotionally brings pains and difficulties to those living with it. Cancer cells remain undifferentiated (continue to divide, causing more damage, and invading new tissue), lack normal cell signaling responses (loss of contact inhibition and evasion of programmed cell death), contain abnormal changes (genetic abnormalities) in chromatin, have altered energy metabolism, and induce vascularization (ensure a steady supply of oxygen and nutrients).

We carefully select 4270 compounds with known anti-tumor activity as Anticancer Active Compound Library that can be used for tumor-related research and anti-tumor drug screening.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L2160

Anti-Cancer Active Compound Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 4270 compounds with known anti-cancer activity for high throughput screening (HTS) and high content screening (HCS);
  • Effective tool for molecular mechanism of tumorigenesis, and anti-tumor drug screening;
  • Covers various major targets including PI3K, HDAC, mTOR, CDK, Aurora Kinase, JAK, etc.
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Packaging And Storage Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
  • This compound library is provided at a concentration of 10 mM in DMSO. A small number of compounds may be provided in different solvents or concentrations due to solubility or stability requirements. Please refer to the specific product information for details.

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Apoptosis
Autophagy
Antibacterial
Endogenous Metabolite
DNA/RNA Synthesis
NF-κB
PI3K
CDK
ROS
EGFR
Ras
VEGFR
Akt
Antibiotic
Parasite
Microtubule Associated
Topoisomerase
Antifungal
mTOR
Caspase
Reactive Oxygen Species
Epigenetic Reader Domain
Bcl-2 Family
Dehydrogenase
Nucleoside Antimetabolite/Analog
COX
FLT
ERK
PDGFR
STAT
Histone Methyltransferase
p38 MAPK
PARP
HDAC
FGFR
Estrogen Receptor/ERR
TNF
c-Met/HGFR
Wnt/beta-catenin
Cytochromes P450
HIV Protease
c-Kit
Ferroptosis
Src
Raf
Interleukin
JAK
MDM-2/p53
Phosphatase
HSP
Antioxidant
MMP
Virus Protease
Influenza Virus
Estrogen/progestogen Receptor
Kras
PKC
Bcr-Abl
AMPK
NO Synthase
ALK
Aurora Kinase
Androgen Receptor
JNK
PPAR
Nrf2
Calcium Channel
E1/E2/E3 Enzyme
P-gp
SARS-CoV
MEK
GSK-3
DUB
TLR
FAK
HIF/HIF Prolyl-Hydroxylase
MAPK
p53
Mitophagy
IL Receptor
PROTACs
DNA Alkylator/Crosslinker
HSV
IGF-1R
TGF-beta/Smad
Mitochondrial Metabolism
Antiviral
AChR
Histone Demethylase
Drug Metabolite
Sirtuin
c-RET
PDE
Chk
Lipoxygenase
ATM/ATR
PERK
Gamma-secretase
Potassium Channel
Proteasome
Tyrosine Kinases
TAM Receptor
HER
Trk receptor
Histone Acetyltransferase
c-Fms
DNA-PK
Pim
Molecular Glues
Cholinesterase (ChE)
Sodium Channel
S6 Kinase
Casein Kinase
Retinoid Receptor
Mdm2
Transferase
Reductase
Adrenergic Receptor
5-HT Receptor
HIF
ROS Kinase
Integrin
Smo
Hedgehog/Smoothened
GABA Receptor
PLK
DNA Methyltransferase
PD-1/PD-L1
ADC Cytotoxin
Serine Protease
IAP
Fatty Acid Synthase
CXCR
Anti-infection
Kinesin
YAP
Histamine Receptor
Aryl Hydrocarbon Receptor
HCV Protease
Glutathione Peroxidase
PKA
HBV
TRP/TRPV Channel
DNA Alkylation
PDK
Tyrosinase
LPL Receptor
c-Myc
Antifolate
Beta Amyloid
GPCR
Dopamine Receptor
Serine/threonin kinase
IDO
Antifection
Isocitrate Dehydrogenase (IDH)
Indoleamine 2,3-Dioxygenase (IDO)
Ligand for E3 Ligase
Phospholipase
S1P Receptor
Carbonic Anhydrase
BTK
DNA
transporter
IκB/IKK
Aromatase
NOS
DHFR
ROCK
MAO
CSF-1R
Immunology/Inflammation related
Prostaglandin Receptor
Syk
IKZF
ATPase
Adenosine Receptor
DYRK
NADPH
Rho
OXPHOS
Monocarboxylate transporter
Photosensitizer
Cell Cycle Arrest
Cysteine Protease
Glutaminase
glycosidase
CaMK
Survivin
AhR
Monoamine Oxidase
IFNAR
Progesterone Receptor
RIP kinase
Glucosidase
Telomerase
BCRP
STING
Ephrin Receptor
Reverse Transcriptase
Proton pump
Amino Acids and Derivatives
Tie-2
GNRH Receptor
Cholecystokinin Receptor
RANKL/RANK
Glucocorticoid Receptor
iGluR
Opioid Receptor
PAK
CCR
Wee1
MNK
PAI-1
Methionine Adenosyltransferase (MAT)
GPX
NOD
IRAK
NOD-like Receptor (NLR)
Chloride channel
MicroRNA
Bcl-6
NAMPT
IRE1
P2X Receptor
ABC Transporter
Somatostatin
Lipid
Acyltransferase
Cannabinoid Receptor
Discoidin Domain Receptor (DDR)
ROR
Ligands for Target Protein for PROTAC
RAAS
Necroptosis
ATG
Liver X Receptor
Leukotriene Receptor
Glucokinase
PYK2
UGT
Endothelin Receptor
Angiotensin-converting Enzyme (ACE)
GluR
Orphan Receptor
PSMA
Aminopeptidase
Pyroptosis
LPA Receptor
BMI-1
HMG-CoA Reductase
Thrombin
p97
PKM
MALT
GTPase
Galectin
Myosin
MTH1
NMDAR
Hexokinase
FAAH
PTEN
cAMP
MELK
p62
Hydroxylase
FOXO
Complement System
Neurokinin receptor
DAPK
NEDD8
CRM1
MyD88
LTR
Arrestin
Lipase
TOPK
Factor Xa
MRP
Serotonin Transporter
FXR
NR4A
GRK
Bombesin Receptor
PAD
Xanthine Oxidase
KSP
Cadherin
Porcupine
CD73
Decarboxylase
ASK
GST
ribosome
KLF
CRISPR/Cas9
Adenosine Deaminase
SGK
Platelet aggregation
APC/C
Protease-activated Receptor
MLK
FOXO3
Thyroid hormone receptor(THR)
RAR/RXR
Factor VIIa
MIF
CaSR
Hck
Neurotensin Receptor
Vitamin
Annexin A
FLAP
Adiponectin Receptor
PAFR
Haspin Kinase
Arp2/3 Complex
DNA gyrase
Stearoyl-CoA Desaturase (SCD)
ACK1
Thrombopoietin Receptor
ATP Citrate Lyase
Beta-Secretase
GPCR19
HuR
RSV
Drug-Linker Conjugates for ADC
Hippo pathway
Acetyl-CoA Carboxylase
FKBP
Protease
PI4K
Cuproptosis
Gap Junction Protein
Sigma receptor
Lysosomal Autophagy
CFTR
PARG(Poly(ADP-ribose) Glycohydrolase)
Apelin receptor
Advanced Glycation End Products
Adenylyl Cyclase
CAT
NPC1L1
CD38
CYP19A1
NUDIX hydrolase
Dynamin
Y Box Binding Protein 1
Arginase
P2Y Receptor
Na+/Ca2+ Exchanger
BACE
gp120/CD4
VDA
Melatonin Receptor
OCT
Kisspeptin
AAK1
B7
LIM Kinase
Stemness kinase
LDLR
Amylase
LAG-3
Prolyl Endopeptidase (PREP)
SIK
FABP
LDL
Na-K-Cl cotransporter
GlyT
Monoamine Transporter
PROTAC Linker
DPP-4
Neuropeptide Y Receptor
Thioredoxin
Vasopressin Receptor
HCAR
Epoxide Hydrolase
Transketolase
Target Protein Ligand-Linker Conjugate
SGLT
PGE Synthase
Glutathione reductase
LRRK2
Free radical scavengers
Urea Transporter
GluCls
NEDD4-1
Carboxypeptidase
TMV
Melanocortin Receptor
GHSR
Aquaporin
RXFP receptor
NADPH-oxidase
Tight Junction Protein
Liposome
Glyoxalase
Ferroportin
ADC Linker
Poly(ADP-ribose) Glycohydrolase (PARG)

Keywords