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AKR1C3-IN-1

Name: AKR1C3-IN-1
Brand: TargetMol
SKU: T7406
Price: 30 USD
Availability: InStock
Rating: 5 (10 reviews)

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Catalog No. T7406Cas No. 327092-81-9

AKR1C3-IN-1 is a potent and selective inhibitor of AKR1C3(IC50 of 13 nM).

AKR1C3-IN-1

🥰Excellent

Purity: 98.02%

Catalog No. T7406Cas No. 327092-81-9

AKR1C3-IN-1 is a potent and selective inhibitor of AKR1C3(IC50 of 13 nM).

Pack Size	Price	Availability
10 mg	$31	In Stock
25 mg	$55	In Stock
50 mg	$98	In Stock
100 mg	$160	In Stock
200 mg	$236	In Stock
1 mL x 10 mM (in DMSO)	$30	In Stock

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Batch Information

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Purity:98.02%

Resource Download

COA HNMR LCMS

Product Introduction

Bioactivity

Description	AKR1C3-IN-1 is a potent and selective inhibitor of AKR1C3(IC50 of 13 nM).
Targets&IC50	AKR1C3:13 nM

Chemical Properties

Molecular Weight	317.36
Formula	C₁₆H₁₅NO₄S
Cas No.	327092-81-9
Smiles	OC(=O)c1cccc(c1)S(=O)(=O)N1CCc2ccccc2C1
Relative Density.	1.397 g/cm3 (Predicted)
Color	White
Appearance	Solid

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 100 mg/mL (315.1 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	3.1510 mL	15.7550 mL	31.5100 mL	157.5498 mL
5 mM	0.6302 mL	3.1510 mL	6.3020 mL	31.5100 mL
10 mM	0.3151 mL	1.5755 mL	3.1510 mL	15.7550 mL
20 mM	0.1575 mL	0.7877 mL	1.5755 mL	7.8775 mL
50 mM	0.0630 mL	0.3151 mL	0.6302 mL	3.1510 mL
100 mM	0.0315 mL	0.1575 mL	0.3151 mL	1.5755 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc