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AKR1C3-IN-1

Catalog No. T7406   CAS 327092-81-9
Synonyms: 3-(3,4-二氢-1H-异喹啉-2-磺酰基)-苯甲酸

AKR1C3-IN-1 is a potent and selective inhibitor of AKR1C3(IC50 of 13 nM).

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AKR1C3-IN-1, CAS 327092-81-9
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Purity: 98%
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Biological Description
Chemical Properties
Storage & Solubility Information
Description AKR1C3-IN-1 is a potent and selective inhibitor of AKR1C3(IC50 of 13 nM).
Targets&IC50 AKR1C3:13 nM
Synonyms 3-(3,4-二氢-1H-异喹啉-2-磺酰基)-苯甲酸
Molecular Weight 317.36
Formula C16H15NO4S
CAS No. 327092-81-9

Storage

Powder: -20°C for 3 years

In solvent: -80°C for 2 years

Solubility Information

DMSO: 100 mg/mL (315.10 mM)

( < 1 mg/ml refers to the product slightly soluble or insoluble )

References and Literature

1. Jamieson S M F , Brooke D G , Heinrich D , et al. 3-(3,4-Dihydroisoquinolin-2(1 H )-ylsulfonyl)benzoic Acids: Highly Potent and Selective Inhibitors of the Type 5 17-β-Hydroxysteroid Dehydrogenase AKR1C3[J]. Journal of Medicinal Chemistry, 2012, 55(17):7746-7758.

Related compound libraries

This product is contained In the following compound libraries:
Inhibitor Library Anti-Metabolism Disease Compound Library Anti-Fibrosis Compound Library Bioactive Compound Library

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What is the mass of compound required to make a 10 mM stock solution in 10 ml of water given that the molecular weight of the compound is 197.13 g/mol?
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What volume of a given 10 mM stock solution is required to make 20ml of a 50 μM solution?
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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

AKR1C3-IN-1 327092-81-9 代谢 NADPH AKR-1C3-IN-1 inhibit AKR1C3IN1 AKR1C3 IN 1 Inhibitor inhibitor