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mAChr-in-1

Catalog No. T5476 CAS 119391-56-9

mAChR-IN-1 is muscarinic cholinergic receptor(mAChR) antagonist (IC50=17 nM).

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mAChr-in-1, CAS 119391-56-9

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Purity: 98%

Biological Description

Chemical Properties

Storage & Solubility Information

Description	mAChR-IN-1 is muscarinic cholinergic receptor(mAChR) antagonist (IC50=17 nM).
Targets&IC50	mAChR:17 nM

Molecular Weight	488.369
Formula	C23H25IN2O2
CAS No.	119391-56-9

Storage

Powder: -20°C for 3 years

In solvent: -80°C for 2 years

Solubility Information

DMSO: 52 mg/mL (106.48 mM)

( < 1 mg/ml refers to the product slightly soluble or insoluble )

References and Literature

1. Wilson AA, et al. Synthesis and biological evaluation of [125I]- and [123I]-4-iododexetimide, a potent muscarinic cholinergic receptor antagonist. J Med Chem. 1989 May;32(5):1057-62.

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Method for preparing in vivo formulation：Take μL DMSO master liquid, next add μL PEG300， mix and clarify, next add μL Tween 80，mix and clarify, next add μL ddH₂O, mix and clarify.

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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

mAChr-in-1 119391-56-9 神经科学 AChR Inhibitor mAChR inhibit Muscarinic acetylcholine receptor mAChr in 1 mAChrin1 inhibitor

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