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LPA2 antagonist 1

🥰Excellent
Catalog No. T15786Cas No. 1017606-66-4

LPA2 antagonist 1 is a highly efficient LPA2 antagonist.

LPA2 antagonist 1

LPA2 antagonist 1

🥰Excellent
Purity: 99.85%
Catalog No. T15786Cas No. 1017606-66-4
LPA2 antagonist 1 is a highly efficient LPA2 antagonist.
Pack SizePriceUSA WarehouseGlobal WarehouseQuantity
1 mg$117-In Stock
5 mg$289-In Stock
10 mg$463-In Stock
25 mg$812-In Stock
50 mg$1,160-In Stock
1 mL x 10 mM (in DMSO)$318-In Stock
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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.
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Batch Information

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Purity:99.85%
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COA HNMR HPLC

Product Introduction

Bioactivity
Description
LPA2 antagonist 1 is a highly efficient LPA2 antagonist.
Targets&IC50
LPA2:17 nM
In vitro
LPA2 antagonist 1 inhibits LPA-induced Erk phosphorylation in a concentration-dependent manner.
LPA2 antagonist 1 inhibits the proliferation of HCT-116 colon cancer cells induced by LPA in a dose-dependent manner. [1]
Chemical Properties
Molecular Weight500.47
FormulaC20H23Cl2N5O2S2
Cas No.1017606-66-4
SmilesN([C@H](CN1CCN(S(=O)(=O)C2=CC(Cl)=C(Cl)C=C2)CC1)C)C3=C4C(C(C)=CS4)=NC=N3
Relative Density.1.453 g/cm3 (Predicted)
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
Solubility Information
DMF: 80 mg/mL (159.85 mM), Sonication is recommended.
DMSO: 80 mg/mL (159.85 mM), Sonication is recommended.
Solution Preparation Table
DMF/DMSO
1mg5mg10mg50mg
1 mM1.9981 mL9.9906 mL19.9812 mL99.9061 mL
5 mM0.3996 mL1.9981 mL3.9962 mL19.9812 mL
10 mM0.1998 mL0.9991 mL1.9981 mL9.9906 mL
20 mM0.0999 mL0.4995 mL0.9991 mL4.9953 mL
50 mM0.0400 mL0.1998 mL0.3996 mL1.9981 mL
100 mM0.0200 mL0.0999 mL0.1998 mL0.9991 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
TargetMol | Animal experimentsFor example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH2O. So your working solution concentration is 2 mg/mL。
Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH2OTargetMol | reagent mix well and clarify
For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.
1 Enter information below:
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g
μL
2 Enter the in vivo formulation:
% DMSO
%
% Tween 80
% Saline/PBS/ddH2O

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc

Keywords

LPA-2 antagonist 1LPA2 antagonist 1LPA2
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