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ASN04885796

🥰Excellent
Catalog No. T30163Cas No. 1032892-26-4
Alias AS-N04885796, ASN 04885796, AS N04885796

ASN04885796 (compound IV) is a neuroprotective, specific GPR17 agonist with an EC50=2.27 nM for GPR17-mediated GTPγS binding and can be used to study neurodegenerative diseases such as cerebral ischemia and demyelinating diseases.

ASN04885796

ASN04885796

🥰Excellent
Purity: 95.36%
Catalog No. T30163Alias AS-N04885796, ASN 04885796, AS N04885796Cas No. 1032892-26-4
ASN04885796 (compound IV) is a neuroprotective, specific GPR17 agonist with an EC50=2.27 nM for GPR17-mediated GTPγS binding and can be used to study neurodegenerative diseases such as cerebral ischemia and demyelinating diseases.
Pack SizePriceAvailabilityQuantity
1 mg$210 In Stock
25 mg$1,400 In Stock
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Purity:95.36%
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Product Introduction

Bioactivity
Description
ASN04885796 (compound IV) is a neuroprotective, specific GPR17 agonist with an EC50=2.27 nM for GPR17-mediated GTPγS binding and can be used to study neurodegenerative diseases such as cerebral ischemia and demyelinating diseases.
Targets&IC50
GTPγS binding assay:2.27 nM (EC₅₀)
In vitro
ASN04885796 (compound IV) is a potent GPR17 agonist, exhibiting an EC₅₀ of 2.27 nM in assays measuring GTPγS binding stimulated by GPR17. ASN04885796 possesses neuroprotective effects and serves as a valuable tool for studying neurological disorders[1].
AliasAS-N04885796, ASN 04885796, AS N04885796
Chemical Properties
Molecular Weight517.55
FormulaC28H28FN5O4
Cas No.1032892-26-4
SmilesO=C(NCC1OCCC1)C(C2=CC=C(F)C=C2)N(C(=O)CN3N=NC=4C=CC=CC43)C5=CC=C(OC)C=C5
Relative Density.1.34 g/cm3 (Predicted)
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice./Shipping at ambient temperature.
Solubility Information
DMSO: 80 mg/mL (154.57 mM), Sonication is recommended.
Solution Preparation Table
DMSO
1mg5mg10mg50mg
1 mM1.9322 mL9.6609 mL19.3218 mL96.6090 mL
5 mM0.3864 mL1.9322 mL3.8644 mL19.3218 mL
10 mM0.1932 mL0.9661 mL1.9322 mL9.6609 mL
20 mM0.0966 mL0.4830 mL0.9661 mL4.8305 mL
50 mM0.0386 mL0.1932 mL0.3864 mL1.9322 mL
100 mM0.0193 mL0.0966 mL0.1932 mL0.9661 mL

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Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH2OTargetMol | reagent mix well and clarify
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