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Rivaroxaban-d4
😃Good
Catalog No. T12736Cas No. 1132681-38-9
Alias Rivaroxaban D4, BAY59-7939 D4, BAY 59-7939 D4, BAY 597939 D4
Rivaroxaban-d4 is a deuterated marker of Rivaroxaban for isotopic tracing.Rivaroxaban (BAY 59-7939) is a highly potent and selective direct inhibitor of coagulation factor Xa (FXa), with an IC50 = 0.7 nM and a Ki of 0.4 nM.
Rivaroxaban-d4
😃Good
Catalog No. T12736Alias Rivaroxaban D4, BAY59-7939 D4, BAY 59-7939 D4, BAY 597939 D4Cas No. 1132681-38-9
Rivaroxaban-d4 is a deuterated marker of Rivaroxaban for isotopic tracing.Rivaroxaban (BAY 59-7939) is a highly potent and selective direct inhibitor of coagulation factor Xa (FXa), with an IC50 = 0.7 nM and a Ki of 0.4 nM.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | TBD | 35 days | |
| 5 mg | TBD | 7-10 days |
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Product Introduction
Bioactivity
Chemical Properties
| Description | Rivaroxaban-d4 is a deuterated marker of Rivaroxaban for isotopic tracing.Rivaroxaban (BAY 59-7939) is a highly potent and selective direct inhibitor of coagulation factor Xa (FXa), with an IC50 = 0.7 nM and a Ki of 0.4 nM. |
| Targets&IC50 | FXa:(ki)0.4 nM , FXa:0.7 nM |
| Alias | Rivaroxaban D4, BAY59-7939 D4, BAY 59-7939 D4, BAY 597939 D4 |
| Molecular Weight | 439.91 |
| Formula | C19H18ClN3O5S |
| Cas No. | 1132681-38-9 |
| Smiles | O=C1N(C[C@H](CNC(=O)C=2SC(Cl)=CC2)O1)C3=C(C(=C(C(=C3[2H])[2H])N4C(=O)COCC4)[2H])[2H] |
| Relative Density. | no data available |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | ||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 40 mg/mL (90.93 mM), Sonication is recommended. | ||||||||||||||||||||||||||||||
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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