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PF-06882961

Catalog No. T12431   CAS 2230198-02-2

PF-06882961 is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.

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PF-06882961 Chemical Structure
PF-06882961, CAS 2230198-02-2
Pack Size Availability Price/USD Quantity
1 mg In stock $ 42.00
5 mg In stock $ 91.00
10 mg In stock $ 158.00
25 mg In stock $ 208.00
50 mg In stock $ 266.00
100 mg In stock $ 457.00
1 mL * 10 mM (in DMSO) In stock $ 111.00
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Purity: 99.54%
Purity: 99.08%
Purity: 98.06%
Purity: 95.1%
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Biological Description
Chemical Properties
Storage & Solubility Information
Description PF-06882961 is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.
In vivo PF-06882961 shows mild to moderate damage to the heart, moderate to severe effects on the thymus gland (which helps with managing infection), mild to moderate stomach ulcers at the highest dose level given in the rat[3].
Molecular Weight 555.6
Formula C31H30FN5O4
CAS No. 2230198-02-2

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

Solubility Information

DMSO: 125 mg/mL (224.98 mM), sonification is recommended.

TargetMolReferences and Literature

1. 20th SCI/RSC Medicinal Chemistry Symposium. 2. Méndez M, et al. Design, Synthesis, and Pharmacological Evaluation of Potent Positive Allosteric Modulators of the Glucagon-like Peptide-1 Receptor (GLP-1R). J Med Chem. 2019 Oct 23. 3. POSSIBLE SIDE EFFECTS AND RISKS OF THE STUDY DRUG AND PROCEDURES.

Related compound libraries

This product is contained In the following compound libraries:
Anti-Cancer Clinical Compound Library Anti-Cancer Drug Library Anti-Obesity Compound Library Anti-Metabolism Disease Compound Library NO PAINS Compound Library Drug Repurposing Compound Library Bioactive Compound Library Bioactive Compounds Library Max Anti-Diabetic Compound Library Clinical Compound Library

Related Products

Related compounds with same targets
BETP L-168049 HAEGTFTSDVS acetate Semaglutide GLP-1 receptor agonist 9 citrate Retatrutide sodium salt GLP-1(7-36), amide Avexitide acetate

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Keywords

PF-06882961 2230198-02-2 GPCR/G Protein Glucagon Receptor PF06882961 PF 06882961 inhibitor inhibit

 

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