Powder: -20°C for 3 years | In solvent: -80°C for 1 year
GNE 2861 inhibits PAK4, PAK5, and PAK6 (IC50s: 7.5, 36, 126 nM, respectively). GNE 2861 is a PAK inhibitor that shows group II selectivity.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 36.00 | |
2 mg | In stock | $ 50.00 | |
5 mg | In stock | $ 79.00 | |
10 mg | In stock | $ 133.00 | |
25 mg | In stock | $ 272.00 | |
50 mg | In stock | $ 455.00 | |
100 mg | In stock | $ 672.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 84.00 |
Description | GNE 2861 inhibits PAK4, PAK5, and PAK6 (IC50s: 7.5, 36, 126 nM, respectively). GNE 2861 is a PAK inhibitor that shows group II selectivity. |
Targets&IC50 | PAK4:7.5 nM, PAK6:126 nM, PAK5:36 nM |
In vitro | GNE 2861 is compound 4 in the reference. |
Molecular Weight | 406.48 |
Formula | C22H26N6O2 |
CAS No. | 1394121-05-1 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 99 mg/mL (243.55 mM), Sonification is recommended.
You can also refer to dose conversion for different animals. More
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GNE 2861 1394121-05-1 Cytoskeletal Signaling PAK p21 activated kinases inhibit Inhibitor GNE-2861 GNE2861 inhibitor