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AN3199

Catalog No. T10316   CAS 1187187-10-5

AN3199 is a selective inhibitor of PDE4 with an IC50 of 94.5 nM.

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AN3199 Chemical Structure
AN3199, CAS 1187187-10-5
Pack Size Availability Price/USD Quantity
2 mg In stock $ 38.00
5 mg In stock $ 60.00
10 mg In stock $ 98.00
25 mg In stock $ 197.00
50 mg In stock $ 317.00
100 mg In stock $ 476.00
1 mL * 10 mM (in DMSO) In stock $ 67.00
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Purity: 100%
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Biological Description
Chemical Properties
Storage & Solubility Information
Description AN3199 is a selective inhibitor of PDE4 with an IC50 of 94.5 nM.
Targets&IC50 PDE4:94.5 nM (IC50)
Molecular Weight 327.14
Formula C17H18BNO5
CAS No. 1187187-10-5

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

Solubility Information

DMSO: 90.0 mg/mL (275.1 mM), Sonication is recommended.

TargetMolReferences and Literature

1. Zhang YK, et al. Design and synthesis of boron-containing PDE4 inhibitors using soft-drug strategy for potential dermatologic anti-inflammatory application. Bioorg Med Chem Lett. 2010 Apr 1;20(7):2270-4. 2. Akama Tsutomu, et al. Preparation of boron-containing small molecules as anti-inflammatory agents. From PCT Int. Appl. (2009), WO 2009111676 A2 20090911.

Related compound libraries

This product is contained In the following compound libraries:
Inhibitor Library Bioactive Compounds Library Max Bioactive Compound Library

Related Products

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Ziritaxestat TP-10 Aminophylline Apremilast PF-04822163 FCPR03 4,5-Dimethoxycanthin-6-one TBA-7371

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Keywords

AN3199 1187187-10-5 Metabolism Others PDE AN 3199 AN-3199 inhibitor inhibit

 

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