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Quininib is a selective antagonist of CysLTR1 and CysLTR2, with IC50 values of 1.2 and 52 μM, respectively, exhibiting anti-angiogenic and anti-tumour effects.
Pack Size | Price | Availability | Quantity |
---|---|---|---|
500 μg | $59 | In Stock | |
1 mg | $86 | In Stock | |
5 mg | $208 | In Stock | |
10 mg | $313 | In Stock | |
25 mg | $527 | In Stock | |
50 mg | $749 | In Stock | |
100 mg | $987 | In Stock |
Description | Quininib is a selective antagonist of CysLTR1 and CysLTR2, with IC50 values of 1.2 and 52 μM, respectively, exhibiting anti-angiogenic and anti-tumour effects. |
Targets&IC50 | CysLT1:1.2 μM, CysLT2:52 μM |
Molecular Weight | 247.29 |
Formula | C17H13NO |
Cas No. | 143816-42-6 |
Smiles | C(=C/C1=C(O)C=CC=C1)\C2=NC3=C(C=C2)C=CC=C3 |
Relative Density. | no data available |
Storage | store at low temperature | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature. |
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