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AC-261066

Name: AC-261066
Brand: TargetMol
SKU: T14089
Price: 30 USD
Availability: InStock
Rating: 5 (10 reviews)

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Catalog No. T14089Cas No. 870773-76-5

Alias AC 261066

AC-261066 is an orally available and isoform-selective agonist of RARβ2 with a pEC50 of 8.0.

AC-261066

🥰Excellent

Purity: 99.64%

Catalog No. T14089Alias AC 261066Cas No. 870773-76-5

AC-261066 is an orally available and isoform-selective agonist of RARβ2 with a pEC50 of 8.0.

Pack Size	Price	Availability
1 mg	$30	In Stock
5 mg	$58	In Stock
10 mg	$106	In Stock
25 mg	$238	In Stock
50 mg	$353	In Stock
100 mg	$495	In Stock
1 mL x 10 mM (in DMSO)	$69	In Stock

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Batch Information

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Purity:99.64%

Resource Download

COA HNMR LCMS

Product Introduction

Bioactivity

Description	AC-261066 is an orally available and isoform-selective agonist of RARβ2 with a pEC50 of 8.0.
Targets&IC50	RARβ2:8.0 （pEC50）
Synonyms	AC 261066

Chemical Properties

Molecular Weight	353.41
Formula	C₁₇H₂₀FNO₄S
Cas No.	870773-76-5
Smiles	CCCCOCCOc1nc(sc1C)-c1ccc(C(O)=O)c(F)c1
Relative Density.	1.247 g/cm3 (Predicted)

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 40 mg/mL (113.2 mM), Sonication and heating to 80℃ are recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	2.8296 mL	14.1479 mL	28.2957 mL	141.4787 mL
5 mM	0.5659 mL	2.8296 mL	5.6591 mL	28.2957 mL
10 mM	0.2830 mL	1.4148 mL	2.8296 mL	14.1479 mL
20 mM	0.1415 mL	0.7074 mL	1.4148 mL	7.0739 mL
50 mM	0.0566 mL	0.2830 mL	0.5659 mL	2.8296 mL
100 mM	0.0283 mL	0.1415 mL	0.2830 mL	1.4148 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc