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A 410099.1, amine-Boc hydrochloride

Catalog No. T39919 CAS 2374122-37-7

A 410099.1, amine-Boc hydrochloride is a functionalized IAP ligand and can be used for the synthesis of PROTACs, such as PROTACs targeting BTK (PROTACs 4 and 5).

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A 410099.1, amine-Boc hydrochloride, CAS 2374122-37-7

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Purity: 98%

Biological Description

Chemical Properties

Storage & Solubility Information

Description

A 410099.1, amine-Boc hydrochloride is a functionalized IAP ligand and can be used for the synthesis of PROTACs, such as PROTACs targeting BTK (PROTACs 4 and 5).

Molecular Weight	620.23
Formula	C32H50ClN5O5
CAS No.	2374122-37-7

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 2 years

Solubility Information

( < 1 mg/ml refers to the product slightly soluble or insoluble )

References and Literature

1. Christopher P Tinworth, et al. PROTAC-Mediated Degradation of Bruton's Tyrosine Kinase Is Inhibited by Covalent Binding. ACS Chem Biol.2019 Mar 15;14(3):342-347

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Method for preparing in vivo formulation：Take μL DMSO master liquid, next add μL PEG300， mix and clarify, next add μL Tween 80，mix and clarify, next add μL ddH₂O, mix and clarify.

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What is the mass of compound required to make a 10 mM stock solution in 10 ml of water given that the molecular weight of the compound is 197.13 g/mol?
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

A 410099.1, amine-Boc hydrochloride 2374122-37-7 A 410099.1, amineBoc hydrochloride A 410099.1, amine Boc hydrochloride inhibitor inhibit

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