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Thrombin inhibitor 1

Catalog No. T10081 CAS 855998-46-8

<a href="/target/Thrombin" style="display: inline; color: #c13a36">Thrombin</a> inhibitor 1 is a potent inhibitor of <a href="/target/Thrombin" style="display: inline; color: #c13a36">Thrombin</a> (Ki: 0.66 nM, 2xaPTT=0.43 μM).

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Thrombin inhibitor 1, CAS 855998-46-8

Pack Size	Availability	Price/USD
5 mg	10-12 weeks	$ 1,370.00
50 mg	10-12 weeks	$ 2,780.00
100 mg	10-12 weeks	$ 3,700.00

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Purity: 98%

Biological Description

Chemical Properties

Storage & Solubility Information

Description	Thrombin inhibitor 1 is a potent inhibitor of thrombin (Ki: 0.66 nM, 2xaPTT=0.43 μM).
Targets&IC50	thrombin(ki):ki： 0.66 nM
In vitro	Thrombin inhibitor 1 (Compound 4) is evaluated for its thrombin inhibitory potency and its functional ability to double the activated partial thromboplastin time (2xaPTT) in human plasma (2xaPTT: 0.43 μM).

Molecular Weight	497.32
Formula	C22H20Cl2F2N4O3
CAS No.	855998-46-8

Storage

Powder: -20°C for 3 years

In solvent: -80°C for 2 years

Solubility Information

( < 1 mg/ml refers to the product slightly soluble or insoluble )

References and Literature

1. Nantermet PG, et al. P2 pyridine N-oxide thrombin inhibitors: a novel peptidomimetic scaffold. Bioorg Med Chem Lett. 2005 Jun 2;15(11):2771-5.

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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

Thrombin inhibitor 1 855998-46-8 Proteases/Proteasome Thrombin Inhibitor inhibitor inhibit

Products are chemical reagents for research use only and are not intended for human use. We do not sell to patients.