keep away from moisture
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Men 10376 is a selective antagonist of tachykinin NK-2 receptor. It has a Ki of 4.4 μM for rat small intestine NK-2 receptor.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
500 μg | 35 days | $ 170.00 | |
1 mg | 35 days | $ 296.00 | |
5 mg | 35 days | $ 1,170.00 |
Description | Men 10376 is a selective antagonist of tachykinin NK-2 receptor. It has a Ki of 4.4 μM for rat small intestine NK-2 receptor. |
Targets&IC50 | NK2 receptor (rat small intestine):(ki)4.4 μM |
In vitro | Men 10376 is a selective tachykinin NK-2 receptor (Ki: 4.4 μM). Men 10376 displays no effect on NK-3 receptor (Ki, >10 μM). It also displays low selectivity for NK-1 and NK-3 receptors (Ki, >10 μM)[1]. Men 10376 shows pA2s of 5.66 and 8.08 for NK-1 (guinea-pig ileum) and NK-2 receptors (endothelium-deprived rabbit pulmonary artery). [2]. |
In vivo | Men 10376 (1 and 3 μmol/kg; in rats) antagonizes an enhance in bladder motility produced by the NK-2 receptor agonist [2]. |
Synonyms | Neurokinin-2 receptor antagonist |
Molecular Weight | 1081.22 |
Formula | C57H68N12O10 |
CAS No. | 135306-85-3 |
keep away from moisture
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
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Men 10376 135306-85-3 Cell Cycle/Checkpoint CDK Neurokinin-2 receptor antagonist inhibitor inhibit