Powder: -20°C for 3 years | In solvent: -80°C for 1 year
CMF019 is a potent agonist of the Apelin receptor (APJ) with G protein bias. CMF019 binds to APJ (pKis: 8.58, 8.49, and 8.71 for the human, rat, and mouse).
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 122.00 | |
5 mg | In stock | $ 259.00 | |
10 mg | In stock | $ 438.00 | |
25 mg | In stock | $ 713.00 | |
50 mg | In stock | $ 985.00 | |
100 mg | In stock | $ 1,320.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 258.00 |
Description | CMF019 is a potent agonist of the Apelin receptor (APJ) with G protein bias. CMF019 binds to APJ (pKis: 8.58, 8.49, and 8.71 for the human, rat, and mouse). |
Targets&IC50 | Apelin receptor (human):pki:8.58 , Apelin receptor (rat):8.49 (pki), Apelin receptor (mouse):8.71(pki) |
Molecular Weight | 455.61 |
Formula | C25H33N3O3S |
CAS No. | 1586787-08-7 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 45 mg/mL (98.8 mM), Sonification is recommended.
You can also refer to dose conversion for different animals. More
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
CMF019 1586787-08-7 GPCR/G Protein Apelin receptor CMF 019 CMF-019 inhibitor inhibit