Powder: -20°C for 3 years
In solvent: -80°C for 2 years
Argipressin is a peptide hormone with vasoconstrictive and antidiuretic activities that binds to the vascular arginine <a href="/target/Vasopressin_Receptor" style="display: inline; color: #c13a36">Vasopressin Receptor</a>, V1, with Kd values of 1.31 and 1.44 nM in A7r5 rat aortic smooth muscle cells and neonatal rat cardiomyocytes, respectively.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In Stock (ship within 1 week) | $ 46.00 | |
2 mg | In Stock (ship within 1 week) | $ 58.00 | |
5 mg | In Stock (ship within 1 week) | $ 91.00 | |
10 mg | In Stock (ship within 1 week) | $ 120.00 | |
25 mg | In Stock (ship within 1 week) | $ 159.00 | |
50 mg | In Stock (ship within 1 week) | $ 189.00 |
Description | Argipressin is a peptide hormone with vasoconstrictive and antidiuretic activities that binds to the vascular arginine vasopressin receptor, V1, with Kd values of 1.31 and 1.44 nM in A7r5 rat aortic smooth muscle cells and neonatal rat cardiomyocytes, respectively. |
In vitro | Argipressin stimulates the intracellular release of calcium in A7r5 cells (EC50 = 5 nM)[1]. |
In vivo | In rat models, argipressin induces hypertension and tachycardia when injected into the lateral septal nuclei at a dose of 100-400 ng and increases heart rate and mean arterial pressure (MAP) when injected into the medial amygdaloid body at a dose of 150-600 ng. |
Synonyms | Arg8-vasopressin, AVP, Vasopressin |
Molecular Weight | 1144.29 |
Formula | C48H69N15O14S2 |
CAS No. | 113-79-1 |
Powder: -20°C for 3 years
In solvent: -80°C for 2 years
H2O: 100 mg/mL (92.23 mM)
( < 1 mg/ml refers to the product slightly soluble or insoluble )
You can also refer to dose conversion for different animals. More
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Argipressin 113-79-1 GPCR/G Protein Vasopressin Receptor Arg8-vasopressin Inhibitor inhibit AVP Vasopressin inhibitor