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Adenosine receptor A1 antagonist 5
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Catalog No. T22466Cas No. 85872-53-3
Adenosine receptor A1 antagonist 5 acts as an adenosine antagonist, is an oxypurine, acts as an insecticide and pest control agent, and has an inhibitory effect on elevated blood pressure.
Adenosine receptor A1 antagonist 5
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Purity: 99.97%
Catalog No. T22466Cas No. 85872-53-3
Adenosine receptor A1 antagonist 5 acts as an adenosine antagonist, is an oxypurine, acts as an insecticide and pest control agent, and has an inhibitory effect on elevated blood pressure.
| Pack Size | Price | USA Warehouse | Global Warehouse | Quantity |
|---|---|---|---|---|
| 1 mg | $41 | In Stock | In Stock | |
| 5 mg | $100 | In Stock | In Stock | |
| 10 mg | $147 | In Stock | In Stock | |
| 25 mg | $252 | In Stock | In Stock | |
| 50 mg | $359 | In Stock | In Stock | |
| 100 mg | $496 | In Stock | In Stock | |
| 200 mg | $667 | - | In Stock |
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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]
This molecule is a custom-made product. TargetMol has an excellent synthesis team with the experience and capability to provide you with cost-effective products.If you have any questions, please feel free to contact us. We are committed to serving you wholeheartedly.
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.
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Purity:99.97%
Appearance:Solid
Color:White
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Product Introduction
Adenosine receptor A1 antagonist 5 AI Summary
Adenosine receptor A1 antagonist 5 exhibits bioactivity primarily as a ligand for adenosine receptors, displaying high binding affinity for the A1 adenosine receptor (Ki = 2.75 nM in rat cortex) and moderate binding affinity for the A2A adenosine receptor (Ki = 116.0 nM in rat striatal membranes). It also shows significant binding affinity for the human HEK293 adenosine A2B receptor (Ki = 18.9 nM). The compound acts as an antagonist at these receptors, inhibiting adenyl cyclase stimulation in various membranes, such as human platelet and rat PC12 membranes, with Ki values indicating a preference for A1 receptors over A2 receptors. Additionally, Adenosine receptor A1 antagonist 5 demonstrates a range of bioactivities, including inhibition of [3H]-PIA binding at adenosine A1 receptors, antagonism at both adenosine A1 and A2 receptors, and inhibition of adenylate cyclase stimulation. Beyond its role in adenosine receptor interaction, the compound shows diverse activity across various biological targets, including inhibitory effects on SARS-CoV-2 cytotoxicity, inhibition of HSD17B4 and JMJD2E, antiviral properties against Lassa and Marburg viruses, and modulation of Cytochrome P450 enzymes..
Note: Summary generated by AI. Data source: ChEMBL 
Bioactivity
Chemical Properties
Storage & Solubility Information
| Description | Adenosine receptor A1 antagonist 5 acts as an adenosine antagonist, is an oxypurine, acts as an insecticide and pest control agent, and has an inhibitory effect on elevated blood pressure. |
| Molecular Weight | 312.37 |
| Formula | C17H20N4O2 |
| Cas No. | 85872-53-3 |
| Smiles | C(CC)N1C2=C(NC(=N2)C3=CC=CC=C3)C(=O)N(CCC)C1=O |
| Relative Density. | 1.218g/cm3 |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature. | ||||||||||||||||||||||||||||||
| Solubility Information | Ethanol: 4.5 mg/mL (14.41 mM), Sonication is recommended. DMSO: 8 mg/mL (25.61 mM), Sonication is recommended.  | ||||||||||||||||||||||||||||||
Solution Preparation Table | |||||||||||||||||||||||||||||||
Ethanol/DMSO
DMSO
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Calculator
In Vivo Formulation Calculator (Clear solution)
Please enter your animal experiment information in the following box and click Calculate to obtain the stock solution preparation method and in vivo formula preparation method:
For example, if the intended dosage is 10 mg/kg for animals weighing 20 g , with a dosing volume of 100 μL per animal, and a total of 10 animals are to be administered, using a formulation of 
10% DMSO+ 40% PEG300+ 5% Tween 80+ 45% Saline/PBS/ddH2O , the resulting working solution concentration would be 2 mg/mL.Stock Solution Preparation:
Dissolve 2 mg of the compound in 100 μL DMSO to obtain a stock solution at a concentration of 20 mg/mL . If the required concentration exceeds the compound's known solubility, please contact us for technical support before proceeding.
Preparation of the In Vivo Formulation:
1) Add 100 μL of the DMSO stock solution to 400 μL PEG300 and mix thoroughly until the solution becomes clear.
2) Add 50 μL Tween 80 and mix well until fully clarified.
3) Add 450 μL Saline,PBS or ddH2O and mix thoroughly until a homogeneous solution is obtained.
This example is provided solely to demonstrate the use of the In Vivo Formulation Calculator and does not constitute a recommended formulation for any specific compound. Please select an appropriate dissolution and formulation strategy based on your experimental model and route of administration.
Dose Conversion
You can also refer to dose conversion for different animals. More Dose Conversion
Tech Support
Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc
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