Powder: -20°C for 3 years
In solvent: -80°C for 2 years
(Rac)-BMS-816336 (Compound 6n) is a racemate of BMS-816336. (Rac)-BMS-816336 is a potent human and mouse 11β-hydroxysteroid <a href="/target/Dehydrogenase" style="display: inline; color: #c13a36">Dehydrogenase</a> type 1 (11β-HSD1) enzyme inhibitor with IC 50 s of 10 nM and 68 nM, respectively. (Rac)-BMS-816336 has good metabolic stability [1].
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
50 mg | 12-16 weeks | $ 1,487.00 | |
100 mg | 12-16 weeks | $ 2,388.00 |
Description | (Rac)-BMS-816336 (Compound 6n) is a racemate of BMS-816336. (Rac)-BMS-816336 is a potent human and mouse 11β-hydroxysteroid dehydrogenase type 1 (11β-HSD1) enzyme inhibitor with IC 50 s of 10 nM and 68 nM, respectively. (Rac)-BMS-816336 has good metabolic stability [1]. |
Targets&IC50 | mouse 11β-HSD1:68 nM , human 11β-HSD1:10 nM |
In vivo | (Rac)-BMS-816336 (compound 6n) has good metabolic stability with the remaining rates in human, mouse and rats of 88%,82% and 72%, respectively [1]. |
Molecular Weight | 341.44 |
Formula | C21H27NO3 |
CAS No. | T12663 |
Powder: -20°C for 3 years
In solvent: -80°C for 2 years
( < 1 mg/ml refers to the product slightly soluble or insoluble )
You can also refer to dose conversion for different animals. More
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(Rac)-BMS-816336 T12663 Metabolism Dehydrogenase (Rac)BMS816336 (Rac) BMS 816336 Inhibitor inhibitor inhibit