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Perzinfotel (Synonyms: EAA-090)

Name: Perzinfotel
Brand: TargetMol
SKU: T16473
Price: 74 USD
Availability: InStock
Rating: 5 (10 reviews)

Catalog No. T16473 Copy Product Info

Purity: 98.35%

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Perzinfotel (EAA-090) is a potent, selective NMDA receptor antagonist (IC50 = 34 nM). It exhibits neuroprotective and analgesic activities, used for stroke and neuropathic pain research.

Perzinfotel

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🥰Excellent

Catalog No. T16473

Synonyms EAA-090

Perzinfotel (EAA-090) is a potent, selective NMDA receptor antagonist (IC50 = 34 nM). It exhibits neuroprotective and analgesic activities, used for stroke and neuropathic pain research.

Cas No. 144912-63-0

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Pack Size	Price	USA Stock	Global Stock
1 mg	$74	-	In Stock
5 mg	$179	-	In Stock
10 mg	$286	-	In Stock
25 mg	$615	-	In Stock
50 mg	$963	-	In Stock
1 mL x 10 mM (in DMSO)	$196	-	In Stock

For In stock only · Estimated delivery: USA Stock (1-2 days) Global Stock (5-7 days)

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Custom-made molecule. TargetMol’s expert synthesis team delivers cost-effective solutions. Contact us for inquiries. Committed to serving you.

For research use only—not for human use. No sales to individuals. Use as intended only.

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Purity:98.35%

Appearance:Solid

Color:Yellow

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COA LCMS HNMR

Product Introduction

Bioactivity

Description	Perzinfotel (EAA-090) is a potent, selective NMDA receptor antagonist (IC50 = 34 nM). It exhibits neuroprotective and analgesic activities, used for stroke and neuropathic pain research.
Targets&IC50	NMDAR:30 nM
In vitro	Perzinfotel dose-dependently blocks NMDA-induced currents (IC50 = 0.48 uM) and protects neurons from glutamate toxicity [1][2].
In vivo	Perzinfotel alleviates chemically induced thermal hypersensitivity and provides analgesia/neuroprotection via selective NMDA binding [1].
Synonyms	EAA-090

Chemical Properties

Molecular Weight	260.18
Formula	C₉H₁₃N₂O₅P
Cas No.	144912-63-0
Smiles	O=C1C(=O)C2=C1NCCCN2CCP(=O)(O)O
Relative Density.	1.60 g/cm3 (Predicted)

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 16 mg/mL (61.5 mM), Sonication is recommmended.

H2O: 4.7 mg/mL (18.06 mM), Sonication is recommmended.

Solution Preparation Table

H2O/DMSO

	1mg	5mg	10mg	50mg
1 mM	3.8435 mL	19.2175 mL	38.4349 mL	192.1746 mL
5 mM	0.7687 mL	3.8435 mL	7.6870 mL	38.4349 mL
10 mM	0.3843 mL	1.9217 mL	3.8435 mL	19.2175 mL

DMSO

	1mg	5mg	10mg	50mg
20 mM	0.1922 mL	0.9609 mL	1.9217 mL	9.6087 mL
50 mM	0.0769 mL	0.3843 mL	0.7687 mL	3.8435 mL

Note : The dilution table applies only to solid products. For liquid products, please calculate the stock solution based on the stated concentration and/or density.

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the stock solution preparation method and in vivo formula preparation method:

For example, if the intended dosage is 10 mg/kg for animals weighing 20 g , with a dosing volume of 100 μL per animal, TargetMol | Animal experiments

and a total of 10 animals are to be administered, using a formulation of TargetMol | reagent

10% DMSO+ 40% PEG300+ 5% Tween 80+ 45% Saline/PBS/ddH₂O , the resulting working solution concentration would be 2 mg/mL.

Stock Solution Preparation:

Dissolve 2 mg of the compound in 100 μL DMSO TargetMol | reagent to obtain a stock solution at a concentration of 20 mg/mL . If the required concentration exceeds the compound's known solubility, please contact us for technical support before proceeding.

Preparation of the In Vivo Formulation:

1) Add 100 μL of the DMSO TargetMol | reagent stock solution to 400 μL PEG300 and mix thoroughly until the solution becomes clear.

2) Add 50 μL Tween 80 and mix well until fully clarified.

3) Add 450 μL Saline,PBS or ddH₂O TargetMol | reagent and mix thoroughly until a homogeneous solution is obtained.

This example is provided solely to demonstrate the use of the In Vivo Formulation Calculator and does not constitute a recommended formulation for any specific compound. Please select an appropriate dissolution and formulation strategy based on your experimental model and route of administration.

All co-solvents required for this protocol, includingDMSO, PEG300/PEG400, Tween 80, SBE-β-CD, and Corn oil, are available for purchase on the TargetMol website.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc