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Opipramol (Ensidon) is an atypical tricyclic antidepressant (TCA) primarily functioning as a sigma (σ) receptor agonist. It interacts effectively with sigma recognition sites, having a Ki value of 50 nM. Opipramol is applicable in the study of generalized anxiety disorder (GAD).
Pack Size | Price | Availability | Quantity |
---|---|---|---|
10 mg | Inquiry | 10-14 weeks | |
50 mg | Inquiry | 10-14 weeks |
Description | Opipramol (Ensidon) is an atypical tricyclic antidepressant (TCA) primarily functioning as a sigma (σ) receptor agonist. It interacts effectively with sigma recognition sites, having a Ki value of 50 nM. Opipramol is applicable in the study of generalized anxiety disorder (GAD). |
In vitro | Opipramol inhibits the uptake of [^3H]DA in crude synaptosomal preparations, with an IC50 value of 5.5 μM [1]. |
In vivo | Opipramol (i.p.; 5-50 mg/kg) has been shown to enhance the release of dopamine in vivo [2]. |
Alias | Opipramol dihydrochloride, G-33040 dihydrochloride, Ensidon dihydrochloride |
Molecular Weight | 436.418 |
Formula | C23H31Cl2N3O |
Cas No. | 909-39-7 |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice./Shipping at ambient temperature. |
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