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Opipramol dihydrochloride

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Catalog No. T204660Cas No. 909-39-7
Alias Opipramol dihydrochloride, G-33040 dihydrochloride, Ensidon dihydrochloride

Opipramol (Ensidon) is an atypical tricyclic antidepressant (TCA) primarily functioning as a sigma (σ) receptor agonist. It interacts effectively with sigma recognition sites, having a Ki value of 50 nM. Opipramol is applicable in the study of generalized anxiety disorder (GAD).

Opipramol dihydrochloride

Opipramol dihydrochloride

😃Good
Catalog No. T204660Alias Opipramol dihydrochloride, G-33040 dihydrochloride, Ensidon dihydrochlorideCas No. 909-39-7
Opipramol (Ensidon) is an atypical tricyclic antidepressant (TCA) primarily functioning as a sigma (σ) receptor agonist. It interacts effectively with sigma recognition sites, having a Ki value of 50 nM. Opipramol is applicable in the study of generalized anxiety disorder (GAD).
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10 mgInquiry10-14 weeks
50 mgInquiry10-14 weeks
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Product Introduction

Bioactivity
Description
Opipramol (Ensidon) is an atypical tricyclic antidepressant (TCA) primarily functioning as a sigma (σ) receptor agonist. It interacts effectively with sigma recognition sites, having a Ki value of 50 nM. Opipramol is applicable in the study of generalized anxiety disorder (GAD).
In vitro
Opipramol inhibits the uptake of [^3H]DA in crude synaptosomal preparations, with an IC50 value of 5.5 μM [1].
In vivo
Opipramol (i.p.; 5-50 mg/kg) has been shown to enhance the release of dopamine in vivo [2].
AliasOpipramol dihydrochloride, G-33040 dihydrochloride, Ensidon dihydrochloride
Chemical Properties
Molecular Weight436.418
FormulaC23H31Cl2N3O
Cas No.909-39-7
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice./Shipping at ambient temperature.

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Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH2OTargetMol | reagent mix well and clarify
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